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2-(2-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
methyl (2S)-3-methyl-2-{[1-(4-methylquinazolin-2-yl)piperidin-4-yl]formamido}butanoate
4-[2-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]-1,2,3,6-tetrahydropyridazine-3,6-dione
methyl (2R,4S)-4-hydroxy-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidine-2-carboxylate
1-ethyl-3-[2-oxo-2-(4-propylpiperazin-1-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
6-({4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]piperidin-4-yl}oxy)quinoline
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-3-phenylpropan-1-one
3-[(4-methyl-1,4-diazepan-1-yl)sulfonyl]-N-(oxan-4-yl)benzamide
6-(4-cyclopentylpiperazin-1-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-[(3R,4S)-1-acetyl-4-phenylpyrrolidin-3-yl]-2-(4-hydroxypiperidin-1-yl)acetamide
1'-(dimethyl-1,3-thiazole-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(2R,3R)-1'-(1-methylcyclohexanecarbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-(1,2-oxazinan-2-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
1-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-3-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]urea
2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-N-(thiophen-2-ylmethyl)acetamide
(4aR,7aS)-1-(3-methylbutanoyl)-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4R)-3-hydroxy-1-(4-hydroxy-1-methylpiperidine-4-carbonyl)piperidin-4-yl]pyridine-4-carboxamide
3-(5-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
4-(3-phenylpropyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[(2,3-dimethoxyphenyl)methyl]-4-[4-(3-methylthiophene-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-[3-(2-aminoethyl)piperidin-1-yl]-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
(2S)-N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyrrolidine-2-carboxamide
4-methyl-2-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenol
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[3-(pyridin-3-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
[(dimethyl-1,3-thiazol-5-yl)methyl][(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
2-butyl-1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-2,5-dihydro-1H-pyrrole
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(quinolin-6-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-3-methylpentane-1,2-dione
1-(6-hydroxy-1,4-oxazepan-4-yl)-3-{[5-(pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}propan-1-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(1,3-thiazol-2-ylmethyl)acetamide
N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N,5-dimethyl-N-[2-(2-oxopiperidin-1-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
4-chloro-1-methyl-3-[1-methyl-3-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
2-(1-benzylpiperidin-4-yl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
3-methyl-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
5-(4-carboxybutanoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-propyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-5-carboxamide
(4aS,7aR)-1-(3-hydroxybenzoyl)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-4-fluoro-N-(furan-2-ylmethyl)benzamide
N-methyl-N-{1-[1-(oxolane-3-carbonyl)piperidin-4-yl]-2-phenylethyl}thiophene-2-carboxamide
N-[(5-chloro-2-ethoxyphenyl)methyl]-N-methyl-3-(1H-pyrazol-1-yl)benzamide
N-methyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(oxan-4-yl)ethyl]acetamide
2-[2-(dimethylamino)ethyl]-9-(2,6-dimethylpyridin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-ethyl-3-{1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
{[2-(azocan-1-yl)pyridin-3-yl]methyl}[(6-methylpyridin-2-yl)methyl]amine
3-(2-chlorophenyl)-3-{2-[4-(2-hydroxyphenyl)piperazin-1-yl]-2-oxoethyl}-1-methylpyrrolidine-2,5-dione
ethyl 1-[(2,5-dimethylphenyl)methyl]-4-(2-methoxyethyl)piperidine-4-carboxylate
(3aR,6aS)-1-oxo-5-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid