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2-(1H-1,3-benzodiazol-1-yl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
2-[(furan-3-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
8-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(4-chlorophenyl)methyl]-N-(1H-imidazol-2-ylmethyl)benzamide
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)cyclobutanamine
[1-(2-fluorophenyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl]dimethylamine
N'-(3-chloro-4-methylphenyl)-N-[2-(1H-imidazol-4-yl)ethyl]propanediamide
1'-(3-ethoxybenzoyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
1-[(3,4-dimethylphenyl)methyl]-4-(1-methyl-1H-pyrazole-4-carbonyl)piperazin-2-one
methyl 4-({[4-(pyridin-3-yl)pyrimidin-2-yl]amino}methyl)benzoate
1-(2-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}-2-oxoethyl)azepan-2-one
3-acetyl-N-ethyl-N-[2-(3-methylphenoxy)ethyl]benzamide
3-(4-hydroxyphenyl)-N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]propanamide
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(1-propylcyclopropyl)acetamide
(3aS,6aS)-2-cyclopentyl-5-[2-(2,3-difluorophenyl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[(4aS,8aR)-1-butyl-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}-1H-pyrazole-3-carboxylic acid
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
5-oxo-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)pyrrolidine-2-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-[4-(1H-imidazol-1-yl)benzoyl]-3-methylpiperidine
3-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-ol
1-(3-methoxyphenyl)-4-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-2-one
5-{2-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-3-(oxolane-2-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
4-[(3,4-dimethoxyphenyl)methyl]-7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-(phenoxathiin-4-yl)-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1S,4S)-2-[2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carbonyl]-2-azabicyclo[2.2.1]heptane
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-{[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]methyl}-6-methylquinolin-4-ol
N-[3-(2-methoxyphenyl)propyl]-1H-indole-3-carboxamide
1-methoxy-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decan-2-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-fluoro-5-sulfamoylbenzamide
3-({[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]carbamoyl}amino)-N-cyclopropyl-4-methoxybenzamide
2-{2-[4-(3,5-dichloro-4-methylbenzoyl)piperazin-1-yl]ethoxy}ethan-1-ol
4-(4-ethyl-1H-pyrazol-5-yl)-1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidine
1-(oxolan-2-ylmethyl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-4-methylpyrimidin-2-amine
4-ethenyl-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylbenzamide
2-amino-7-hydroxy-4-[4-(2-hydroxyethoxy)phenyl]-5H-indeno[1,2-b]pyridine-3-carbonitrile
1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-(diethylamino)-1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
N-{[1-(3-acetamidopropanoyl)piperidin-3-yl]methyl}-3,5-dimethoxybenzamide
2-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)-1H-1,3-benzodiazole
N4-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-6-(propan-2-yl)pyrimidine-2,4-diamine
3-[2-chloro-5-(morpholin-4-yl)phenyl]-1-[(1-ethylpiperidin-2-yl)methyl]urea
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(2,5-dimethylphenyl)methyl]pyrrolidine-2-carboxylate
2-phenyl-1-{1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidin-4-yl}ethan-1-ol
1-benzyl-8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 3-({1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazol-4-yl}formamido)propanoate