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5-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
3-(2-methoxybenzoyl)-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidine
2-amino-4-[2-(2-hydroxyethoxy)phenyl]-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(1S,6R)-9-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
[2-({imidazo[1,2-a]pyrimidin-6-ylmethyl}(thiophen-3-ylmethyl)amino)ethyl]dimethylamine
5-[1-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,4-dimethylbenzamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(3,4-dimethoxyphenyl)methyl]propanamide
(2E)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
[4-({1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-(2-{4-[({[4-(difluoromethoxy)phenyl]methyl}(methyl)amino)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)methanesulfonamide
4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-ethylpiperidine-1-carboxamide
1-(3-methylbutyl)-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
1-(4-{[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}piperazin-1-yl)-2,2-dimethylpropan-1-one
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
1-(2-methoxy-5-{[methyl(oxan-4-yl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
2-hydroxy-5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)benzoic acid
4-(oxolan-3-yl)-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-1,2,3-triazole
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
[(3R,5R)-1-(5-methyl-1,3,4-thiadiazol-2-yl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
(1R,3S)-3-amino-N-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)cyclohexane-1-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}pyrrolidine-2-carboxamide
1-[2-(dimethylamino)ethyl]-6-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-(pyridin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-({5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazol-3-yl}formamido)acetamide
(3S,4R)-4-(3-fluorophenyl)-1-{[4-(2-hydroxyethoxy)phenyl]methyl}pyrrolidine-3-carboxylic acid
N-[1-(7-{[3-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]methanesulfonamide
1-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(1,3-thiazol-4-yl)ethan-1-one
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-1,2,5-thiadiazole-3-carboxamide
N-(3-hydroxypropyl)-3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]propanamide
2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(1-hydroxypropan-2-yl)acetamide
methyl 2-[N-methyl-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamido]acetate
3-{[(2S)-1-hydroxy-3-methylbutan-2-yl]sulfamoyl}-N-(pyrimidin-4-ylmethyl)benzamide
1-[4-(furan-2-carbonyl)piperazin-1-yl]-2-(morpholin-3-yl)ethan-1-one
2-[(3,4-dimethoxyphenyl)methyl]-N-(2-hydroxyethyl)-N-methyl-1,3-benzoxazole-6-carboxamide
(1S,5R)-N-(furan-2-ylmethyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
5,7-dimethyl-N-[(4-methyl-1,4-oxazepan-6-yl)methyl]pyrido[2,3-d]pyrimidin-4-amine
1-[3-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-oxopropyl]pyrrolidin-2-one
(3aR,5S,6S,7aS)-2-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-octahydro-1H-isoindole-5,6-diol
5-(3-methylbutyl)-5-[1-(2-phenylacetyl)piperidin-4-yl]-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
6-chloro-N,N-dimethyl-3-{[methyl(quinolin-4-ylmethyl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-(2-{[5-(3,4-difluorophenoxymethyl)-1,2-oxazol-3-yl]formamido}ethyl)acetamide
(4aS,8aR)-6-[(2E)-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
(3R,5R)-N-(2-methylpropyl)-1-(naphthalen-2-ylmethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
methyl 2-[(2-phenylethyl)sulfamoyl]-6-(1,3-thiazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-methyl-N-[1-(pyridin-2-yl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N,N-dimethyl-2-[(1S,5R)-3-(6-methylpyridine-3-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide