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1-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-3-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)urea
methyl (2S,4R)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-[3-(3-fluorophenyl)benzamido]pyrrolidine-2-carboxylate
N-[2-(dimethylamino)ethyl]-5-(4-fluoro-3-methylbenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
ethyl 4-({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amino)piperidine-1-carboxylate
(3R,4R)-1-[(2-benzoyl-1-benzofuran-3-yl)methyl]-4-ethylpiperidine-3,4-diol
1-(carbamoylmethyl)-N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-3-carboxamide
2-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}-4-methoxyphenol
3,3,3-trifluoro-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}propanamide
(1S,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(2,3-dichlorophenyl)-5-(methanesulfonylmethyl)pyridine
2-(4-butyl-2,3-dioxopiperazin-1-yl)-2-phenyl-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
({4-[1-(cyclohexylmethyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-yl}methyl)dimethylamine
3-[(1-acetylpiperidin-4-yl)oxy]-N-cycloheptyl-4-methoxybenzamide
1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-diazepane
(4aR,8aS)-1-[2-(diethylamino)ethyl]-6-(thiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
(3S,4S)-3-hydroxy-N-(2-methyl-1H-1,3-benzodiazol-6-yl)-4-(propan-2-yloxy)pyrrolidine-1-carboxamide
3-[3-(4-methanesulfonylphenyl)phenyl]-1H-pyrazole
(4S)-3,3,4-trimethyl-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
1-ethyl-8-{[3-(furan-2-yl)phenyl]methyl}-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(pyridin-3-ylmethyl)piperidin-4-yl]oxy}benzamide
N-[(4-fluorophenyl)methyl]-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methylacetamide
(2S,4S)-N-ethyl-4-[2-(2-ethyl-1H-imidazol-1-yl)acetamido]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
2-{[2-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}quinolin-4-ol
2-(4-methoxyphenoxymethyl)-N-methyl-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
2-(5-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(2-chlorophenyl)ethyl]propanamide
ethyl 1-[6-(1-benzothiophen-3-yl)-3-(morpholine-4-carbonyl)pyridin-2-yl]piperidine-3-carboxylate
2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-(propan-2-yl)-1H-imidazole
5-cyclobutanecarbonyl-1'-[(4-methyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclopropyl-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperazine-2-carboxamide
2-{3-methyl-5-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-ethyl-1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperidine-3-carboxylic acid
2-{3-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]propyl}-5-fluoro-1H-1,3-benzodiazole
2-{4-[2-(4-fluorophenoxy)ethyl]phenyl}acetamide
5-chloro-3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
4,6-dimethyl-1-{3-oxo-3-[4-(oxolan-2-ylmethyl)piperazin-1-yl]propyl}-1,2-dihydropyrimidin-2-one
1-(2-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)methyl]acetamide
N-({7-[2-(4-chloro-2-methylphenoxy)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-fluorobenzamide
8-(5-ethenylpyridin-2-yl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopropyl-2-(dimethylamino)-2-(2-fluorophenyl)-N-(pyridin-2-ylmethyl)acetamide
4-{5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
2-{1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
5-[(1S,2R)-2-butylcyclopropanecarbonyl]-3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-N,N-dimethylmorpholine-2-carboxamide
N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-(thiophene-3-carbonyl)piperidine-3-carboxamide
(2S)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]-3-(pyridin-4-yl)propanoic acid