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2-(2-chloro-5-methylphenyl)-N-ethylpyrimidin-4-amine
1-{1-[(2E)-4-methylpent-2-enoyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-methyl-N-[1-(1-{spiro[2.4]heptane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
2-[(3-ethoxy-2-hydroxypropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-[1-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)cyclohex-3-ene-1-carboxamide
1-(4,6-dimethylquinazolin-2-yl)-N-(oxan-4-ylmethyl)piperidine-4-carboxamide
(1R,3S)-7-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-7-azaspiro[3.5]nonane-1,3-diol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[4-(1H-pyrazol-4-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
7-(2-hydroxyethyl)-2-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-{2-[3-(2-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-methoxy-4-[4-(4-methoxyphenyl)butan-2-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl N-{1-oxo-1-[3-oxo-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-8-yl]propan-2-yl}carbamate
2-methoxy-N-{2-[3-(morpholin-4-ylmethyl)phenoxy]propyl}acetamide
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
methyl (2S,4R)-4-hydroxy-1-({4-[(5-methyl-1,3,4-thiadiazol-2-yl)carbamoyl]phenyl}methyl)pyrrolidine-2-carboxylate
3-{[(1H-imidazol-2-ylmethyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-hydroxy-N-[2-(2-hydroxyethoxy)ethyl]-2-phenylpyrimidine-5-carboxamide
N,N-dimethyl-3-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]aniline
6-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-1,3-benzothiazole
1-(4,7-dimethylquinazolin-2-yl)-N-[(4-methoxyphenyl)methyl]azepan-4-amine
N-[2-hydroxy-3-(piperazin-1-yl)propyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
(1R,9S)-5-amino-12-methyl-3-[2-(piperidin-1-yl)pyrimidin-5-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
5-acetyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}thiophene-3-carboxamide
ethyl 4-(cyclopropylmethyl)-1-[(2-methoxyphenyl)methyl]piperidine-4-carboxylate
N-(2-{7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-(4-fluorophenyl)acetamide
2-ethyl-1-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
N-{4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}acetamide
{4-[(4-chlorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methanol
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
8-(5-chloropyridin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[3-(4-methylpiperazin-1-yl)propyl]-6-(propan-2-yl)pyrimidin-4-amine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-methyl-2-(morpholin-4-yl)-N-[2-(propylsulfanyl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(thiophen-2-yl)propan-1-one
ethyl 3-{[7-(pyridine-4-amido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]amino}propanoate
6-methyl-1-[2-(methylsulfanyl)phenyl]-4-(pyridine-4-carbonyl)piperazin-2-one
methyl 3-{6-[(3-methoxyphenyl)methoxy]-2-oxo-4-[3-(thiophen-2-yl)propanoyl]-1,4-diazepan-1-yl}propanoate
N3-(2-hydroxyethyl)-N1,N1-dimethyl-N3-[(4-methylphenyl)methyl]piperidine-1,3-dicarboxamide
[(2-ethoxypyridin-3-yl)methyl]({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
N-cyclopropyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(3-chlorobenzoyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
6-(2,5-dimethylfuran-3-yl)-2-[3-(hydroxymethyl)piperidine-1-carbonyl]-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})(pyridin-3-ylmethyl)amine
N-(2-methoxyethyl)-1,3-dimethyl-2,6-dioxo-N-(thiophen-2-ylmethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
ethyl 1-[2-(morpholin-4-yl)-6-phenylpyridine-3-carbonyl]piperidine-2-carboxylate
3-[({6,7-dimethoxy-1-[(4-methylphenyl)methyl]-2-oxo-1,2-dihydroquinolin-3-yl}methyl)amino]-1λ6-thiolane-1,1-dione
8-[(2-aminopyridin-3-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one