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N-{4-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]-4-oxobutyl}acetamide
8-(2,3-dimethylbenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(3-methoxypropyl)-1-[2-methyl-5-(trifluoromethyl)benzoyl]piperidine
(3S,4S)-4-cyclopropyl-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidine-3-carboxylic acid
1-(4-benzylpiperazin-1-yl)-3-{1-[(2,4-difluorophenyl)methyl]piperidin-3-yl}propan-1-one
3-(2-fluorophenyl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-2-(pyridin-4-yl)acetamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-[4-(pyrrolidin-1-yl)benzoyl]pyrrolidin-3-amine
2-[(2-hydroxy-2-phenylethyl)amino]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]-3-(3-fluorophenyl)-1-methylpyrrolidine-2,5-dione
7-methyl-4-[(6-methylpyridin-2-yl)methyl]-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[2-(1H-imidazol-4-yl)ethyl]-2-(4-methyl-1H-imidazol-5-yl)-1H-imidazole
6-ethyl-2-methyl-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]quinoline
7-methyl-2-{2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
N-[(2R,3R)-1'-[(2,5-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
(2R)-2-({2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)propanamide
1,5-dimethyl-4-{[3-(3-phenylpropanoyl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
1-[(1-hydroxycyclohexyl)methyl]-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
1-(cyclohexylmethyl)-N-methyl-6-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
methyl 3-[(2-ethylbutanamido)methyl]-5-[3-(trifluoromethyl)benzamido]benzoate
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide
3-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-1-(2-methoxyethyl)-1-(1,3-thiazol-2-ylmethyl)urea
2-(pyridin-2-ylsulfanyl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
1-(3-{4-[4-(propan-2-yl)-1,4-diazepan-1-yl]piperidin-1-yl}phenyl)pyrrolidin-2-one
8-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-[2-(4-phenylpiperidin-1-yl)ethyl]-1-(pyridin-3-yl)urea
2-{2-[3-hydroxy-3-(hydroxymethyl)pyrrolidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
N-[(2,3-dimethoxyphenyl)methyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-[(4aR,8aS)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
7-(2-hydroxyethyl)-2-{[2-(propylamino)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-({1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)thiophene-2-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-1-(pyrimidin-2-yl)piperidin-4-amine
(2S,4R)-4-butanamido-N,N-diethyl-1-(2-methylbenzoyl)pyrrolidine-2-carboxamide
2-(furan-3-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
1-[(3-hydroxyphenyl)methyl]-3-propylpiperidine-3-carboxylic acid
diethyl({[1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]methyl}sulfamoyl)amine
6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(4aR,8aS)-1-[2-(diethylamino)ethyl]-6-[4-(3-fluorophenyl)benzoyl]-decahydro-1,6-naphthyridin-2-one
1-{1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-4-yl}-2-phenylethan-1-ol
2-[4-(1,3-dihydroxypropan-2-yl)-6-hydroxy-1,4-diazepan-1-yl]pyridine-4-carbonitrile
1-{2-[({4-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-3-methoxyphenyl}methyl)amino]ethyl}piperidin-2-one
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(3-{[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
N-methyl-2-(3-methylbutanoyl)-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
6-methoxy-N,3-dimethyl-N-[3-(oxolan-2-yl)propyl]-1-benzofuran-2-carboxamide
3-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-3-yl)-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-(5-cyano-1,3-thiazol-2-yl)-4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}benzamide
2-methyl-2-{4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]phenyl}propanenitrile
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-(ethylamino)-N-methylpyrimidine-5-carboxamide
methyl 6-(2,2-dimethylpropyl)-2-[(4-fluorophenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(4aR,7aS)-1-(2-benzyl-1,3-thiazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione