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1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(2-phenylethyl)piperidin-3-yl]piperazine
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-[(dimethylcarbamoyl)methyl]piperazine-1-carboxamide
N5-butyl-1-cyclohexyl-N3-methyl-N3-[(1-methylpiperidin-3-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(methoxymethyl)-1-[1-(naphthalene-1-sulfonyl)piperidin-4-yl]-5-(trifluoromethyl)-1H-1,3-benzodiazole
N-{2-[(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}phenyl)formamido]ethyl}acetamide
3-(4-cyclohexylphenyl)-1-methyl-1-(oxan-4-yl)urea
N-({1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)-1H-indole-2-carboxamide
methyl(oxolan-2-ylmethyl){[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
[4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)morpholin-2-yl]methanamine
methyl (2S,4S,5R)-5-(2,3-difluorophenyl)-4-[(2,2-dimethylpropyl)carbamoyl]-1-methylpyrrolidine-2-carboxylate
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
N-[(2R,3R)-1'-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-(dimethylamino)-2-{4-[(1-methyl-1H-indol-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
1-(2H-1,3-benzodioxol-4-ylmethyl)-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
methyl 1-[(3S,5S)-1-benzyl-5-[(quinolin-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-(4-phenylazepane-1-carbonyl)-N-(pyridin-3-ylmethyl)pyridin-2-amine
2-{4-[(3,5-dimethyl-1H-indol-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
methyl 6-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]benzamide
3-[3-(hydroxymethyl)quinolin-2-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
4-{4-[(1S,5S)-3-azabicyclo[3.3.1]nonane-3-carbonyl]phenyl}-2-methylbutan-2-ol
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
(2S)-2-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}-3-phenylpropanamide
5-({1-[2-(1H-imidazol-5-yl)ethyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl}methyl)-2-methyl-1H-1,3-benzodiazole
5-[4-(2-ethylmorpholine-4-carbonyl)-6,8-dimethylquinolin-2-yl]pyrimidin-2-amine
(1S,5R)-3-(pyridin-2-ylmethyl)-6-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-[1-(furan-2-ylmethyl)piperidin-3-yl]-3-phenylpropan-1-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N,6-dimethyl-2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
(1S,5R)-3-(2-methoxypyridine-3-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-(4-fluorophenyl)-N-(2-hydroxybutyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
9-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]sulfonyl}-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
N-[2-(2,4-difluorophenyl)-1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
1'-(4-chloro-3-fluorobenzoyl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-methylpyrimidin-2-amine
1-(2-methoxy-4-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
1-(1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
1,3-dimethyl-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-pyrazole-5-carboxamide
1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(piperidin-1-yl)piperidine
1-{4-[1-(cyclopent-3-en-1-yl)-4-phenyl-1H-imidazol-5-yl]phenyl}ethan-1-one
N-[1-(4-chlorophenyl)ethyl]-2-(4-ethylpiperazin-1-yl)acetamide
N-cyclohexyl-3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carboxamide
N-[2-(2-chloro-6-fluorophenyl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
5-(1-cyclobutanecarbonylpiperidin-4-yl)-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
3-(3-fluoro-4-phenylbenzoyl)-N-(propan-2-yl)piperidine-1-carboxamide
3-methyl-6-{[3-(pyridin-2-yl)azetidin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
3-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(2-methyl-5-propanamidophenyl)piperidine-1-carboxamide