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4-(4-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenyl)-2-methylbutan-2-ol
1-(2-aminoethyl)-N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
5-ethyl-5-{1-[(2-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
7-cyclobutaneamido-N-[(2,5-difluorophenyl)methyl]-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2-{[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}phenol
2-{3-[2-(methylsulfanyl)ethyl]-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
3-(3-methoxyquinoxalin-2-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
methyl 2-(diethylsulfamoyl)-6-(2,4,5-trifluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(but-2-yn-1-yl)-5-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
4-methyl-2-{2-[4-phenyl-5-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-6-(trifluoromethyl)pyrimidine
(2E)-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-3-yl)prop-2-enamide
2-(dimethylamino)-N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(4-methylphenyl)acetamide
2-(3-chloro-4-hydroxyphenyl)-N-[3-(pyridin-4-yl)propyl]acetamide
2-methyl-2-({2-methyl-3-[(pyridin-3-ylmethyl)amino]phenyl}formamido)propanoic acid
1-(2-{1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
(3R,4S)-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-4-phenylpyrrolidin-3-amine
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-5-phenyl-1,2-oxazole-3-carboxamide
(2S)-2-amino-3-cyclohexyl-N-[2-(dimethylsulfamoyl)ethyl]propanamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)furan-2-carboxamide
1-{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}-4-(oxolane-2-carbonyl)piperazine
{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
[(3R,4R)-1-(pyridin-4-ylmethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-methyl-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-1,3-thiazole-4-carboxamide
5-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]pyridine-2-carbonitrile
1-phenyl-N-({1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}methyl)methanesulfonamide
9-(2-hydroxyacetyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(2-ethylpyridine-4-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
{[1-({1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methyl}(methyl)amine
6-(2-chloro-4-fluorophenyl)pyridin-2-amine
4-[2-(benzylamino)pyrimidin-5-yl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(3-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenyl)-6-(oxolan-3-yl)-3,4-dihydropyrimidin-4-one
1-[2-(benzyloxy)ethyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(propan-2-ylsulfanyl)acetyl]-1,4-diazepan-5-one
{3-[(2-fluorophenyl)methyl]-1-(3-methoxy-4-methylbenzoyl)piperidin-3-yl}methanol
(3S,4R)-1-[3-(pyridin-2-yl)propanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-cyclopentyl-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-(2-chloro-4-fluorophenoxymethyl)-N-[(3S)-2-oxoazepan-3-yl]-1,2-oxazole-3-carboxamide
4-({3-[3-(diethylamino)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)piperazin-2-one
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-2-cyclopentyl-N-(2-methoxyethyl)-2-phenylacetamide
(2S,4R)-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-(4-fluorophenyl)-3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carboxamide
N-({3-[(dimethylamino)methyl]phenyl}methyl)-2-(4-methoxyphenyl)acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
4-(4-{[2-(2,4-dimethoxyphenyl)ethyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
2-methyl-4-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3-thiazole-5-carboxamide
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
6-fluoro-2-{[(2-hydroxy-2-phenylethyl)amino]methyl}quinolin-4-ol
3-methyl-5-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-2-yl)-1,2-oxazole
2-(4-fluorophenyl)-2-hydroxy-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}acetamide