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2-[5-(2,3-dimethoxyphenyl)-3-methyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-(cyclopropylmethyl)-4-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-2-(propan-2-yl)-1,4-diazepane
[3-(2-phenylethyl)-1-(quinoxalin-2-yl)piperidin-3-yl]methanol
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-[1-(pyridin-2-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(3-chlorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(1-ethyl-1H-pyrazole-4-carbonyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
4-(4-methoxyphenyl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}butanamide
methyl 2-(benzylsulfamoyl)-6-[(4-methylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-fluorobenzamide
1-[2-({[3-(cyclopentyloxy)phenyl]carbamoyl}amino)ethyl]piperidine-3-carboxamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-benzothiophene-5-carboxamide
1-(5-propyl-1,2-oxazole-4-carbonyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N-[(3R,4S)-1-(2-chloro-3-methylbenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
9-(2-hydroxy-3-methylbutanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]urea
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1H-imidazole-5-carboxamide
3-(2-chlorophenyl)-3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-1-(3-methoxypropyl)pyrrolidine-2,5-dione
2-[({1-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}oxy)methyl]pyridine
{[4-(1-{imidazo[1,2-a]pyridine-3-carbonyl}piperidin-2-yl)phenyl]methyl}dimethylamine
4-tert-butyl-2-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-ylmethyl}phenol
4-[(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]oxane-4-carbonitrile
2-(3-{3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}-5-methyl-1H-pyrazol-1-yl)-N-methylacetamide
3-(2-oxo-2-{4-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)-4-(2-phenylethyl)piperazin-2-one
1-benzyl-8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopentyl-5-(4-methyl-1,3-oxazole-5-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[4-(methylsulfanyl)benzoyl]pyrrolidin-3-yl]methanol
2-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
1-{2-methyl-4-[({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-phenylmethanesulfonylbenzamide
1-acetyl-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]piperidine-3-carboxamide
2-(2-aminoethyl)-5,6-dimethyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
N-[(3-chloro-4-methoxyphenyl)methyl]-N-methylthian-4-amine
3-hexyl-8-(oxolane-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
6-[(3S,4S)-3-(azepan-1-yl)-4-hydroxypyrrolidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
4-(2-methylquinolin-4-yl)-N-[2-(pyridin-4-yl)ethyl]morpholine-2-carboxamide
methyl (1R,3S,3aR,6aS)-3-[4-methoxy-3-(prop-2-en-1-yl)phenyl]-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-6-methyl-2-oxo-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(quinolin-5-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-methoxy-3-[(4-methyl-1H-imidazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
4-[(4-chlorophenyl)methyl]-3-[(4-hydroxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
(2S,4R)-4-amino-1-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-hydroxy-3-methoxy-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}benzamide
2-(1-methyl-1H-imidazol-2-yl)-1-(1-phenylbutyl)-1H-imidazole
3-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chlorophenyl)urea
2-cyclopropyl-N-[(2-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide