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N-{2-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
4-[(2-fluorophenyl)methyl]-1-[(2-methoxyphenyl)methyl]-1,4-diazepan-5-one
1-(carbamoylmethyl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}piperidine-3-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
methyl 3-acetamido-1-ethyl-5-{[(3-hydroxy-4-methoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-ethyl-4-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}piperazine-2,3-dione
2-{2-[1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
1-[3-(pyrazin-2-yl)propanoyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
1-(morpholin-4-yl)-3-[1-(quinoxaline-6-carbonyl)piperidin-4-yl]propan-1-one
N-butyl-3-[(3-methoxyphenyl)methyl]-N-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(3-hydroxyphenyl)-4-oxo-4-[4-(pyridin-4-yl)piperidin-1-yl]butanamide
1-cyclopropyl-N-(2-methylpropyl)-6-oxopiperidine-3-carboxamide
(3aR,6aS)-5-[4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carbonyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-{3-[3-(morpholine-4-carbonyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-ethyl-3-methyl-3-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidine
4-(4-chlorophenyl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methylbutanamide
(3R,4S)-4-cyclopropyl-1-(furan-2-ylmethyl)-N,N-dimethylpyrrolidin-3-amine
(2S,4R)-4-(benzylamino)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-(cyclohexylmethyl)-N,N-dimethyl-5-[(propan-2-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-{1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}-2-methoxyphenol
5-[({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-{[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]amino}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
N-(1-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylfuran-3-carboxamide
2-fluoro-N-({8-[2-(7-methyl-2-oxo-2H-chromen-4-yl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
1-cyclohexyl-4-[(2,6-difluorophenyl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-(pyridin-3-yl)-4-{[4-(trifluoromethyl)phenyl]methyl}piperazine
4-(2-hydroxyethyl)-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]piperazine-1-carboxamide
1-(2-amino-6-methylpyrimidine-4-carbonyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
2-(2,4,6-trimethylphenyl)pyridine-4-carboxamide
N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
N-(4,6-dimethylpyridin-2-yl)-3-[(3-acetamidopyrrolidin-1-yl)methyl]benzamide
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-amino-N-cyclopropyl-4-methyl-N-[(3-methylthiophen-2-yl)methyl]-1,3-benzothiazole-6-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(methylsulfanyl)propanamide
N-[2-(dimethylamino)ethyl]-7-methyl-N-[(5-methylthiophen-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
methyl 9-(cyclopentyloxy)-7-oxo-3-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1R,5S,8S)-3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-8-methoxy-3-azabicyclo[3.2.1]octane
diethyl({[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}sulfamoyl)amine
1-cyclopentanecarbonyl-N-methyl-N-[1-(pyridin-3-yl)propyl]piperidine-4-carboxamide
8-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
4-[(2-methylpyridin-3-yl)oxy]-N-[1-(pyridin-4-yl)propan-2-yl]piperidine-4-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-methyl-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
N-cyclopentyl-4-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-oxopentanamide
5-(3-methylbut-2-en-1-yl)-1'-(pyridin-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{[4-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}(methyl)[2-(pyridin-2-yl)ethyl]amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-3-yl)piperazine
7-[(2,3-difluorophenyl)methyl]-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decane