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methyl({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(propan-2-yl)amine
(4aR,7aS)-1-(2-methylpropyl)-4-(6-oxo-1,6-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(methoxymethyl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)thiophene-2-carboxamide
2-(3-methoxyphenyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
1-(cyclohexylmethyl)-N-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-amine
({4-ethyl-5-[1-(3-methoxybenzoyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
5-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
2-[methyl(quinoxalin-2-ylmethyl)amino]-N-[2-methyl-6-(propan-2-yl)phenyl]acetamide
1-ethyl-4-[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]pyrrolidin-2-one
(2S,4R)-4-acetamido-N,N-diethyl-1-(4-fluoro-2-methylbenzoyl)pyrrolidine-2-carboxamide
(2S,4S)-1-benzyl-N-methyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-(7-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-2-(methylamino)pyridine-4-carboxamide
1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
2-[(dimethylcarbamoyl)amino]-N-methyl-N-[(4-phenoxyphenyl)methyl]acetamide
N-(1-{1-[4-(dimethylamino)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N'-[3-(dimethylamino)-1-phenylpropyl]-N-(2-ethoxyphenyl)propanediamide
4-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1-ethyl-3,5-dimethyl-1H-pyrazole
3-[2-oxo-2-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethyl]imidazolidine-2,4-dione
2-butyl-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[2-methoxy-5-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
7-(3-chlorophenyl)-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-oxopyrrolidin-1-yl)benzamide
methyl 5-(cyclohexylamino)-3-acetamido-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-chloro-4-({1-[1-(4-fluorophenyl)propan-2-yl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
1,4-dimethyl 2-[(1-{4-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]phenyl}piperidin-4-yl)amino]butanedioate
ethyl 5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(3R,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
1-(furan-3-ylmethyl)-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
5-[(4-fluorophenyl)methyl]-3-(oxan-4-ylmethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
4-[3-methyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N-methyl-1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-amine
3-(2-methoxyethyl)-1-[3-(2-methylphenyl)propanoyl]piperidine-3-carboxylic acid
3-(5-{2-[methyl(1-methylpiperidin-4-yl)amino]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
1-(furan-3-ylmethyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
7-chloro-2-(2-cyclopropylpyrimidin-5-yl)-4-(piperidine-1-carbonyl)quinoline
N-(3-methylphenyl)-3-{1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-4-yl}propanamide
2-(2-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}phenoxy)ethan-1-ol
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(2-methoxyethyl)-1H-pyrazole-4-carboxamide
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine-3-carboxylate
1-(4-cyclohexylpiperazin-1-yl)-4-(1H-pyrazol-4-yl)butan-1-one
methyl N-{2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}carbamate
4-[7-(5-ethylthiophene-2-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
3-(2,5-dioxoimidazolidin-4-yl)-N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}propanamide
N-methyl-1-(oxolan-2-ylmethyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
7-fluoro-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(2-methylpyrimidin-5-yl)quinoline-4-carboxamide
1-[1,3-dioxo-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-[1-(naphthalen-1-yl)ethyl]piperidine-3-carboxamide
2-methyl-6-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)pyrimidin-4-ol