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4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
3-methyl-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-oxopentanamide
N-(3-cyanothiophen-2-yl)-3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)benzamide
4-acetamido-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
N-(2H-1,3-benzodioxol-5-yl)-1-[4-(piperidin-1-yl)benzoyl]piperidin-3-amine
N-[(3-methyl-1-benzofuran-2-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-benzyl-3-ethylpiperidine-3-carboxylic acid
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-ethyl-4-methyl-1,3-thiazole-5-carboxamide
5-[1-(2-cyclopentyl-2-phenylacetyl)piperidin-4-yl]-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
1-cyclohexyl-4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperazine
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-2-(furan-2-yl)azepane
6-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]-2,3-dihydropyridazin-3-one
methyl 9-(benzyloxy)-3-[(4-fluorophenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
ethyl 1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
6-{4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-9H-purine
4-{1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}-1-(2-methylpropyl)piperidine
[(3,5-dimethoxyphenyl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-[5-(thiophen-2-yl)furan-2-yl]propanamide
[(3S,5R)-1-(2,3-difluoro-4-methylbenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
5-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
1-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}piperidine-3-carboxamide
6-(1-cyclopentylpiperidine-4-carbonyl)-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
3-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
2-(2-ethyl-1H-imidazol-1-yl)-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-indole-6-carboxamide
1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)azepan-4-amine
N-[(2R)-1-hydroxy-3-phenylpropan-2-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
(3S)-N-tert-butyl-2-(1H-imidazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2-methylpiperidine-2-carboxylic acid
2-(4-phenylpiperidin-1-yl)-N-{3-[(pyridin-3-yl)amino]propyl}acetamide
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-2-(methylsulfanyl)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
6-chloro-4-[3-(3-methoxypropyl)piperidine-1-carbonyl]-2-methylquinoline
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
(4aR,7aS)-4-[(2,6-difluorophenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(1S,5R)-3-benzyl-6-{5H,6H-imidazo[2,1-b][1,3]thiazole-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
8-(2,1,3-benzothiadiazol-5-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{4-[(2,3-dihydro-1H-inden-1-yl)amino]piperidin-1-yl}phenyl)-N-[2-(2-methoxyphenyl)ethyl]acetamide
2-(2-{[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-(4-methylpentyl)-4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}morpholine
5-[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1H-pyrrole-3-carbonitrile
(3R,4R)-1-(2,5-dimethylpyrimidin-4-yl)-3,4-dimethylpyrrolidin-3-ol
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-2-(morpholin-4-yl)benzamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(4-phenylphenyl)acetamide
1-(4-{[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]methyl}phenyl)ethan-1-one
2-methoxy-1-(4-{4-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
1-{2-oxo-2-[4-(2-oxo-1,3-oxazolidin-3-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydroquinolin-2-one
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}urea
6-[(diethylamino)methyl]-N-(2-methoxy-2-methylpropyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide