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1-(cyclopropylmethyl)-3-(isoquinolin-5-yl)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
1-(cyclopropylmethyl)-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-2-(propan-2-yl)-1,4-diazepane
N-{2-methyl-1-[7-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}methanesulfonamide
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1-benzoxepine-4-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-{[(4-fluorophenyl)methyl]sulfanyl}propan-1-one
(4aS,8aR)-1-propyl-6-[3-(pyrazin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
3-(3-hydroxy-3-methylbutyl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}benzamide
1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethan-1-one
(3S,4R)-4-(pyridin-3-yl)-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidine-3-carboxylic acid
2-chloro-5-acetamido-N-{imidazo[1,2-a]pyridin-2-ylmethyl}benzamide
5-acetyl-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-2,4-dimethyl-1H-pyrrole-3-carboxamide
4-[(3-methylthiophen-2-yl)methyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[6-(trifluoromethyl)pyridin-2-yl]benzamide
2-[3-(azepan-1-ylmethyl)phenyl]-6-(2-methylpropyl)-3,4-dihydropyrimidin-4-one
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
4-[(2,6-dimethylpyridin-3-yl)oxy]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxylic acid
2-(3-methoxypropyl)-8-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
[5-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)-2-ethoxyphenyl]methanol
methyl 3-cyclopropaneamido-6-{[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
diethyl({2-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]ethyl})amine
(3aS,6aS)-1-(2-cyclopentylacetyl)-N-(thiophen-2-ylmethyl)-octahydropyrrolo[3,4-b]pyrrole-5-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3,4-dimethoxybenzamide
(3S,4R)-1-[2-methyl-2-(morpholin-4-yl)propanoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
methyl 3-benzamido-5-{[2-(2-fluorophenyl)acetamido]methyl}benzoate
3-propyl-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,2-oxazole
4-methoxy-6-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
N-{[4-fluoro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(4-methoxyphenyl)furan-2-carboxamide
5-(azepan-1-yl)-1-benzyl-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({5-[(4-ethoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
3-[({1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}oxy)methyl]pyridine
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-phenylethane-1,2-dione
methyl 6-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2-[(3-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(2-methylpropyl)-N-[3-(methylsulfanyl)propyl]-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-1,2,3-triazole
5-(2-fluoro-3-methoxyphenyl)-1-(2-fluoroethyl)-4-phenyl-1H-imidazole
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
2,6,8-trimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]pyridin-2-amine
6-fluoro-N-methyl-2-oxo-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
methyl 1-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-2-carboxylate
(2S)-2-hydroxy-4-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}butanoic acid
3,5-dimethyl-4-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
1-{3-cyclopropyl-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl}isoquinoline
2-(4-acetylphenoxy)-1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]ethan-1-one
1-(7-fluoro-2-methylquinoline-4-carbonyl)-4-phenylpiperidine-4-carbonitrile
1-(carbamoylmethyl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}piperidine-4-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
5-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione