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7-[(2S,3R)-2-amino-3-hydroxybutanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(2-methoxyethyl)-3-({1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}oxy)benzamide
2-{3-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]phenoxy}acetamide
N-(1-benzylpiperidin-4-yl)-2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-[5-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-(1-benzylpiperidin-4-yl)-N-(3-methylbutyl)piperidine-3-carboxamide
3-chloro-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
5-methyl-5-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}-3-(pyridin-4-ylmethyl)imidazolidine-2,4-dione
N-[(2S)-2-aminopropyl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
3-methyl-7-{[4-(methylsulfanyl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}-1,4-oxazepan-6-ol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(1,4-oxazepan-4-yl)pyridine-3-carboxamide
(2S,4S)-4-amino-1-[(3,5-dichlorophenyl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
N-[2-(azepan-1-yl)-2-phenylethyl]-1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
dimethyl({4-methyl-5-[1-(pyridin-4-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-(3-fluorophenyl)-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
8-(2,3-dihydro-1H-inden-2-yl)-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-cyclohexyl-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(2,2-dimethyloxan-4-yl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
6-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-methylimidazo[1,2-a]pyridine
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-1,2,3-triazol-1-yl)ethan-1-one
ethyl 4-[4-(4-{[2-(pyridin-4-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
1-benzyl-3-(oxolan-3-yl)-5-(5-propyl-1,2-oxazol-3-yl)-1H-1,2,4-triazole
4-(4-fluoro-3-methoxyphenyl)-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(4-methoxy-3-methylphenyl)-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)ethan-1-one
1-[2-methoxy-5-({[(2-methylphenyl)methyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
8-(2-aminoacetyl)-3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(1S,5R)-6-(2-methyl-1-benzofuran-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
methyl 5-{[(2E)-2-methylbut-2-en-1-yl]amino}-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-(2-phenoxyethyl)piperidin-3-yl)methanol
N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylfuran-3-carboxamide
8-(4-methylpyrimidine-5-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-[(3S,4R)-1-(5-methoxy-1H-indazole-3-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
6-fluoro-2-oxo-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-cyclohexyl-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrazole
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidine
2-methyl-N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-(2,5-dimethoxyphenyl)-3-(thiophene-2-sulfonamidomethyl)piperidine-1-carboxamide
2-(1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
4-benzyl-3-ethyl-1-[(2-methoxypyrimidin-5-yl)methyl]-1,4-diazepan-5-one
N-(furan-2-ylmethyl)-3-[2-(3-methoxyphenyl)ethyl]piperidine-1-carboxamide
8-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
3-({2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)-1-(4-methylpiperidin-1-yl)propan-1-one
N,1-dimethyl-N-(quinolin-5-ylmethyl)-1H-pyrrole-2-carboxamide
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
5-{4-[(2,3-dihydro-1H-inden-5-yloxy)methyl]piperidine-1-carbonyl}-2-ethylpyrimidine
[1-(pyrazine-2-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
methyl 2-{[(3-chlorophenyl)methyl]sulfamoyl}-6-propanoyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate