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(4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,4-oxazepan-6-yl)methanol
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propane-1,3-diol
5-methyl-1-(3-methylphenyl)-4-[4-(2-methylpropyl)benzoyl]piperazin-2-one
7-(2-methoxyethyl)-2-(5-propyl-1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,4R)-4-(4-methylphenyl)-1-[3-(pyridin-4-yl)propanoyl]pyrrolidin-3-yl]acetamide
2-(4-{[4-(5-chloro-2-fluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-ol
N4-cyclopropyl-6-(2-ethoxypyridin-3-yl)pyrimidine-2,4-diamine
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-{1-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
2-[(4-chlorophenyl)methyl]-8-[6-(dimethylamino)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
2-(3-hydroxypropyl)-9-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-methanesulfonylphenyl)-5-(2-methyloxolan-2-yl)-3-phenyl-1H-1,2,4-triazole
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)butan-1-one
3-(1-benzyl-5-oxopyrrolidin-3-yl)-4-(naphthalen-1-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidine
methyl[(3-methylpyridin-4-yl)methyl]{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-6-(trifluoromethyl)pyridine-3-carboxamide
4-ethyl-6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-methylpyrimidine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-hydroxyethyl)piperidine-4-carboxamide
8-[(3-hydroxyphenyl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(3-methylbutyl)-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
8-fluoro-2-[3-(2-methylphenoxy)azetidine-1-carbonyl]quinoline
1-[1-(2-phenylethyl)piperidin-4-yl]-N-(piperidin-4-yl)piperidine-3-carboxamide
4-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[(2S)-1-{7-[(2-chloro-6-fluorophenyl)(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
4-[2-methoxy-4-(3-propoxypiperidine-1-carbonyl)phenoxy]-1-methylpiperidine
2,2-dimethyl-6-(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidine-1-carbonyl)-3,4-dihydro-2H-pyran-4-one
2-{[(1-hydroxybutan-2-yl)[(2-methylphenyl)methyl]amino]methyl}-3-methoxyphenol
N-methyl-3-(1,2-oxazinan-2-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}propanamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[2-(pyridin-4-yl)ethyl]propanamide
N-[(3R,4S)-1-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]ethane-1-sulfonamide
N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]-1-phenylcyclohexane-1-carboxamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
(4aS,7aR)-1-(pyridazine-3-carbonyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[(1-ethyl-1H-imidazol-5-yl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
N-{2-[1-(3-methylbut-2-en-1-yl)piperidin-3-yl]ethyl}cyclopropanesulfonamide
3-(methylsulfanyl)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)propan-1-one
ethyl 6-({2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxylate
1-(1,3-oxazole-5-carbonyl)-4-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,4-diazepan-6-ol
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
(2S,4S)-N-ethyl-1-(1,3-thiazol-2-ylmethyl)-4-(thiophene-2-amido)pyrrolidine-2-carboxamide
4-(hydroxymethyl)-1-(5-methyl-2-phenylfuran-3-carbonyl)azepan-4-ol
2-methyl-N-[(2-phenoxypyridin-3-yl)methyl]-1H-1,3-benzodiazole-4-carboxamide
4-{3-[4-chloro-3-(trifluoromethyl)phenyl]-1-methyl-1H-1,2,4-triazol-5-yl}morpholine
ethyl 4-(3-phenylpropyl)-1-[2-(pyridin-3-yl)acetyl]piperidine-4-carboxylate
4-[3-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(2,4-dimethylphenyl)-2-{[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]amino}acetamide
6-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-3-[1-(3-methylbut-2-enoyl)piperidin-3-yl]-N-(1-methylpiperidin-4-yl)propanamide