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11-{[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-benzyl-N,N-dimethyl-5-[(2,2,2-trifluoroethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-benzyl-8-[(2-ethoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(3-chlorophenyl)methyl]-N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-1,3-benzoxazole-6-carboxamide
1-[(3-acetylphenyl)methyl]-4-(3-tert-butyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
1-[(4-methylphenyl)methyl]-4-[3-(morpholin-4-yl)butanoyl]piperazin-2-one
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(5-phenyl-4H-1,2,4-triazol-3-yl)acetamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-(2-oxoazonan-1-yl)acetamide
7-[(2-fluorophenyl)methyl]-2-(4-methyl-1H-imidazole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-[4-(methoxycarbonyl)piperidin-1-yl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(1R,5R)-3-(2-benzyl-1,3-thiazole-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-{[3-methyl-7-(4-phenylbutanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
5-(4-methoxyphenyl)-N-(2-phenylpropyl)-1,2,4-triazin-3-amine
2,4-dichloro-3-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)phenol
3-[1-(1H-indole-2-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
1-{2-[methyl(6-methylhept-5-en-2-yl)amino]ethyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(cyclopropylmethyl)-N-propyl-1,3-oxazole-4-carboxamide
9-methoxy-3-[(4-methoxyphenyl)methyl]-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
8-(2-methoxybenzenesulfonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(3-chlorophenoxy)propan-1-one
N'1-(2-methylpropyl)-N'1-[(3-methylthiophen-2-yl)methyl]cyclopropane-1,1-dicarboxamide
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
1-(3-methoxyphenyl)-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
3-cyclopropyl-1-[(4-ethylphenyl)methyl]-5-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazole
2-(3-methoxyphenyl)-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
(2-methoxyethyl)({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[(4-methylphenyl)methyl]amine
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylpyrimidin-2-amine
1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(2-methylphenyl)-1,4-diazepane
9-[2-(3-methoxyphenyl)acetyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethyl-6-(2-methylpropyl)pyrimidine-4-carboxamide
1-{2-[3-(dimethylamino)pyrrolidin-1-yl]acetyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl({1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-phenylethyl})(pyridin-3-ylmethyl)amine
2-(1-ethyl-1H-pyrazol-4-yl)-6,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)quinoline
2-{[2-(diethylamino)ethyl](ethyl)sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
ethyl 1-(3-fluorophenyl)-5-[({[1-(morpholin-4-yl)cyclopentyl]methyl}amino)methyl]-1H-pyrazole-4-carboxylate
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-3-cyclopropyl-N-methyl-1H-pyrazole-5-carboxamide
6-methyl-4-{9-oxa-2-azaspiro[5.5]undecan-2-yl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(2-propoxyethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[3-(methylsulfanyl)phenyl]methyl})amine
N-[(2-chlorophenyl)methyl]-N-cyclopropyl-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
{1-[(2-chlorophenyl)methyl]-3-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
N-[(3R,4S)-1-[(4-methoxypiperidin-1-yl)sulfonyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-(4-chlorophenyl)-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutane-1-carboxamide
2-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}quinoxaline
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]propanamide
(3R,4R)-4-cyclopropyl-3-methyl-1-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]piperidin-4-ol
5-methoxy-2-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol