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(3R,4R)-1-(5-chlorofuran-2-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
4-({4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)benzoic acid
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(1-cyclopentylpiperidin-3-yl)methyl]-4-methyl-N-[2-(piperidin-1-yl)ethyl]-1,2,5-oxadiazole-3-carboxamide
{2-[(1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]ethyl}dimethylamine
1-[2-(dimethylamino)ethyl]-4-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}pyrrolidin-2-one
N-[(2R,3R)-1'-(5-methylthiophene-2-carbonyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
{3-[(4-fluorophenyl)methyl]-1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl}methanol
(5S,9aS,9bS)-5-(1-benzofuran-2-yl)-2-(2,3-dihydro-1H-inden-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(2-chlorophenyl)ethyl]-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-ethyl-5-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]-1,2-oxazole-4-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-{1-[(2-fluorophenyl)methyl]-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
butyl N-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)carbamate
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
1-cyclopentyl-4-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)-1,4-diazepane
5-(4-benzylpiperidin-1-yl)-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-hydroxy-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-(piperidin-4-ylmethyl)-3-(1,3,4-thiadiazol-2-yl)urea
4-(1H-pyrazol-4-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]butanamide
N-[(3R,4S)-1-(cyclopropylmethyl)-4-phenylpyrrolidin-3-yl]-2-methanesulfonamidoacetamide
1-cyclopropyl-N-[3-(4-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide
5-[ethyl(2-methylprop-2-en-1-yl)amino]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
4-[4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]phenol
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-amino-4-{methyl[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]amino}quinazoline-6-carboxylic acid
3-(4-methoxyphenoxymethyl)-1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
2-(3-fluoro-4-methylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-[2-(4-methoxyphenyl)phenyl]-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxamide
N-benzyl[(1H-1,2,3-benzotriazol-5-yl)amino]sulfonamide
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-methylphenyl)ethan-1-one
5-benzenesulfonamido-N-cyclopentyl-1-ethyl-2-methyl-1H-1,3-benzodiazole-7-carboxamide
N-[(2R,3R)-2-methoxy-1'-[(2,3,6-trifluorophenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
5-(2-ethoxypyridin-3-yl)-2-methoxy-4,6-dimethylpyridine-3-carbonitrile
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}amine
3-ethyl-1-(2-phenylethyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-oxo-6-[(4-phenylazepan-1-yl)methyl]-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-(2-hydroxyethyl)-N-[2-(2-methoxyphenyl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-{4-[6-(morpholin-4-yl)pyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
1-[(3-methoxyphenyl)methyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
4-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]butan-1-one
9-methoxy-4-[(4-methylphenyl)methyl]-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-(cyclobutylmethyl)-2-[3-(2-methoxyphenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(3-methylphenyl)acetamide