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4-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1-phenylpiperazin-2-one
2-amino-N-[3-(1,3-benzoxazol-2-yl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
5-(4-aminoquinolin-8-yl)thiophene-2-carboxylic acid
6-({[(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amino}methyl)-1,4-oxazepan-6-ol
2-{[4-(dimethylamino)phenyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(8-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]oxolane-2-carboxamide
[1-({[2-methyl-7-(piperidin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}methyl)cyclobutyl]methanol
3-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-1-{3-[(5-methylpyridin-2-yl)amino]propyl}urea
6-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]quinoline
2-[2-(1H-1,2,3-triazole-5-carbonyl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl]pyridine
1-[3-(aminomethyl)pyrrolidin-1-yl]-2-methyl-2-[(4-methylphenyl)amino]propan-1-one
2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(quinazolin-2-yl)piperazin-1-yl]ethan-1-one
1-methanesulfonyl-4-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperazine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-amino-6-(1-methyl-1H-pyrrol-3-yl)-4-[5-(1H-pyrazol-3-yl)furan-2-yl]pyridine-3-carbonitrile
N-{1-benzyl-7-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazol-5-yl}acetamide
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-(7-methyl-1-benzofuran-2-carbonyl)morpholine
1-benzyl-4-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
4-(6-chloro-2H-1,3-benzodioxol-5-yl)-3-methyl-2-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(2R,3R)-1'-[(3,4-dimethylphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
(1R,3S)-N1-[3-(dimethylamino)-2,2-dimethylpropyl]-N3-ethyl-1,2,2-trimethylcyclopentane-1,3-dicarboxamide
1-benzyl-6-(pyridin-2-ylmethoxy)-4-(1,2,3-thiadiazole-4-carbonyl)-1,4-diazepan-2-one
2-(cyclohex-1-en-1-yl)-N-({5-fluoro-7-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
1-(5-phenyl-1,2-oxazole-4-carbonyl)azepane
methyl (2S)-1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
ethyl 2-(1-{3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanoyl}piperidin-2-yl)acetate
dimethyl({4-methyl-5-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-(2-methoxyacetyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]piperidine-3-carboxamide
N4,N4,5-trimethyl-N2-[1-(1-methyl-1H-pyrazol-5-yl)propyl]pyrimidine-2,4-diamine
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
methyl (2S)-2-{[1-(6-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]amino}-3-methylbutanoate
1-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propan-1-one
N-cyclohexyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-(2-phenylethyl)propanamide
N-{[8-(4-chlorobenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclohexanecarboxamide
N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-4-(pyrrolidin-1-yl)benzamide
1-{4-[(cyclohexylmethyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
3-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propanamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
5-methyl-3-(2-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-2,3-dihydro-1,3-benzoxazol-2-one
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(2-methoxyphenoxy)acetamide
(2S,4R)-4-amino-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-N,N-diethylpyrrolidine-2-carboxamide
4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-1λ6-thiane-1,1-dione
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-2-(methylsulfanyl)pyridine-3-carboxamide
2-cyclopentyl-N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-4-hydroxy-2-methylpyrimidine-5-carboxamide
3-{[(2-hydroxyethyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-{5-[6-amino-5-cyano-4-(5-cyano-1-methyl-1H-pyrrol-3-yl)pyridin-2-yl]thiophen-3-yl}acetic acid