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1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(pyridin-2-yl)propan-1-one
1-ethyl-N-[2-(4-fluorophenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-{[(5-methylfuran-2-yl)methyl]amino}-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(3-methylpyridin-2-yl)methyl]piperidine-3-carboxamide
(4aS,8aR)-6-(furan-3-carbonyl)-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-{[1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
2-ethyl-9-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[1,3-dioxo-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(2-hydroxy-2-phenylethyl)-N-methylpiperidine-4-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3,4-dimethyl-5-sulfamoylbenzamide
(1S,5R)-3-(1-methyl-1H-pyrrole-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
9-methoxy-N-methyl-7-oxo-3-{spiro[2.4]heptane-1-carbonyl}-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(3-chloro-4-methoxyphenyl)-6-(2-methylbenzoyl)-6-azaspiro[2.5]octane-1-carboxamide
ethyl 1-{3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanoyl}piperidine-3-carboxylate
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(2-methylphenoxymethyl)piperidine
3-chloro-4-{[1-(3-cyclopentylpropyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
2-cycloheptyl-1-[4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]ethan-1-one
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
2-[4-(5-acetylthiophen-3-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
N-({5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-[5-({[(2-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
(3R,9aR)-3-benzyl-8-[(3-fluorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N,2-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(1H-pyrazol-1-yl)propanamide
2-chloro-6-methoxy-4-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}phenol
5-({4-[6-(trifluoromethyl)pyridin-2-yl]piperazin-1-yl}methyl)pyrimidin-2-amine
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}acetamide
(1-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-2-phenylethyl)(methyl)(pyridin-3-ylmethyl)amine
N-[2-(2-fluorophenyl)-1-[1-(thiolan-3-yl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
1-{3-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-[2-(dimethylamino)ethyl]-6-oxopiperidine-3-carboxamide
5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-(pyridin-2-ylmethyl)piperidin-2-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-(4-ethylphenyl)-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[(2-ethoxyphenyl)methyl]cyclopropanamine
5-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
5-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-N-ethylpyrimidin-2-amine
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(5-methylfuran-2-yl)methyl]acetamide
ethyl N-{[(3S,4S)-3-hydroxy-1-[(3E)-pent-3-enoyl]piperidin-4-yl]methyl}carbamate
4-(piperidin-1-yl)-1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidine-4-carboxamide
1-methyl-N-[2-(morpholin-4-yl)ethyl]-5-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
9-(2-acetylbenzoyl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-[(1S,5R)-6-[3-(prop-2-en-1-yloxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
6-[(2E)-3-(3,4-dimethoxyphenyl)prop-2-enoyl]-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[(3R,4S)-1-[3-(dimethylamino)pyrazin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-methoxy-2-methylpropanamide
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]acetamide
1-(cyclopropylmethyl)-3-[(2-methylphenyl)methyl]-6-[2-(1H-1,2,3,4-tetrazol-1-yl)pyridine-4-carbonyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(1-{7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide