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2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-N-ethylpyrimidin-2-amine
N-[(2R,3R)-1'-[(2-fluoro-4-methoxyphenyl)methyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
3-[(3R,4S)-4-(dimethylamino)-1-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]piperidin-3-yl]propanoic acid
3-phenyl-1-(1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)propan-1-ol
3-(4-methyl-1,3-thiazol-5-yl)-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]propanamide
2-[1-(2-methanesulfonylethyl)-1H-1,2,3-triazol-4-yl]-1-(prop-2-en-1-yl)-1H-1,3-benzodiazole
methyl 3-[(2-fluorophenyl)methyl]-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}propan-1-one
6-[(4-fluorophenyl)methoxy]-4-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-1-(propan-2-yl)-1,4-diazepan-2-one
methyl 3-{[1-(cyclopropylmethyl)-5-(2-fluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
1-(2-hydroxyethyl)-5-(1-phenylcyclopentanecarbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[2-({[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}amino)pyrimidin-4-yl]pyrrolidin-3-ol
2-benzyl-9-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-chloro-5-(1H-pyrazol-1-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]benzamide
1-[3-(3-fluorophenyl)benzoyl]-4-(pyrrolidin-3-yl)piperazine
4-(5-methyl-1,2-oxazole-3-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3,5-dimethoxy-N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)benzamide
2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[1-(thiophen-2-yl)propan-2-yl]acetamide
methyl 3-(furan-2-amido)-1-methyl-5-[(oxan-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]amine
(2S,4R)-4-amino-N-ethyl-1-{2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}pyrrolidine-2-carboxamide
2-(3,4-dimethoxyphenyl)-5-fluoro-1-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
6-(2,6-dimethylhept-5-en-1-yl)-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
4-methyl-N-[2-(5-methylthiophen-2-yl)ethyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-[1-tert-butyl-5-(1H-pyrazol-3-yl)-1H-1,2,4-triazol-3-yl]pyridine
2-ethyl-1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine
4-(cyclohexylmethyl)-3-[1-(propan-2-yloxy)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{2,7-dimethylpyrazolo[1,5-a]pyrimidin-5-yl}-3-(2-phenylethyl)-1H-1,2,4-triazole
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 6-(2-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
7-(2-methylphenyl)-4-[(2R)-pyrrolidine-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[(butan-2-yl)amino]-N-cyclopentyl-5-(phenylsulfamoyl)benzamide
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-[(4-phenyloxan-4-yl)methyl]acetamide
2-ethyl-4-methyl-N-[(5-methylpyrazin-2-yl)methyl]-1,3-oxazole-5-carboxamide
2-{[(4-methylpyrimidin-2-yl)amino]methyl}-3,4-dihydroquinazolin-4-one
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
2-[(2-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}phenyl)amino]acetic acid
(3R,4S)-1-(2,6-dimethylpyrimidine-4-carbonyl)-3,4-dimethylpiperidin-4-ol
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-amido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(2-hydroxybutyl)sulfamoyl]benzamide
N-(1-methylpiperidin-4-yl)-2-(morpholin-4-yl)-N-(2-phenylethyl)butanamide
methyl 1-[(3S,5S)-1-[(2,5-dimethylphenyl)methyl]-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(4-{[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}phenoxy)ethan-1-ol
7-methoxy-1-methyl-2-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-[(3-methoxyphenyl)methyl]-N-methyl-N-[(4-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-methyl-N-[2-(2-methylphenyl)-1-{1-[2-(piperidin-1-yl)acetyl]piperidin-4-yl}ethyl]-2-(1H-pyrazol-1-yl)acetamide