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N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(thiophen-3-yl)acetamide
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
(4aR,8aS)-1-[2-(diethylamino)ethyl]-6-[3-(3-fluorophenyl)benzoyl]-decahydro-1,6-naphthyridin-2-one
4-(1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidine-3-carbonyl)morpholine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methylpiperidine-2-carboxamide
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-(2,4-dimethoxyphenyl)propanamide
N-cyclopropyl-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pyridine-4-carboxamide
3-chloro-N-(morpholin-2-ylmethyl)-5-(trifluoromethyl)pyridin-2-amine
4-(2,6-dimethylpyridin-4-yl)-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]piperazine-1-carboxamide
N-cyclopropyl-1-{1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]piperidin-4-yl}piperidine-4-carboxamide
N-(1-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
N-[2-chloro-5-(2-methoxyacetamido)phenyl]-6-hydroxy-1,4-oxazepane-4-carboxamide
2-cyclobutyl-5-(2-methoxyacetamido)-1-methyl-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methoxymethyl)piperidine
N-[(3S,4R)-1-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]-4-propylpyrrolidin-3-yl]acetamide
4-[(3-chlorophenyl)methyl]-1-(quinolin-8-ylmethyl)-1,4-diazepan-5-one
1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
2-(4-methyl-1H-imidazol-5-yl)-1-[2-(oxolan-2-ylmethoxy)phenyl]-1H-imidazole
1-[cyclohexyl(methyl)amino]-3-(3-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
ethyl 1-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperidine-2-carboxylate
1-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydroquinoxalin-2-one
1-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
5-(4-fluorophenyl)-N-[2-(oxolan-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[2-(dimethylamino)ethyl]-6-methyl-3-(3-methylpiperidine-1-carbonyl)-2-(2-phenylethyl)-1,4-dihydropyridin-4-one
N-(2-ethoxyethyl)-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}[2-(pyridin-3-yloxy)ethyl]amine
6-(3-chloro-4-fluorobenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-(naphthalen-1-yl)ethyl]propanamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(6-methylpyridin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]methanesulfonamide
3-({2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazol-5-yl}formamido)propanoic acid
N,3,4,7-tetramethyl-N-(1H-pyrazol-3-ylmethyl)-1H-indole-2-carboxamide
5-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]pyrazin-2-ol
(1R,5R)-N,N-dimethyl-6-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-methyl-2-[4-(piperidin-1-yl)piperidin-1-yl]quinazoline
1-({1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-yl}amino)propan-2-ol
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)piperidine-3-carboxylate
2-methyl-1-(4-{methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}piperidin-1-yl)propan-1-one
5-[(2-methoxyethyl)amino]-1-methyl-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 6-{[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]methyl}-3-propanamidothieno[2,3-b]pyridine-2-carboxylate
({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
9-[(2S)-2-amino-2-benzylpropanoyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-methyl-1H-1,2,3-benzotriazole-4-sulfonamide
N-[(2-aminopyrimidin-5-yl)methyl]-6-ethyl-N,2-dimethylquinoline-4-carboxamide
1-{[2-(2-phenylethoxy)phenyl]methyl}-1,4-diazepan-5-one
1-{2-[4-phenyl-5-(quinolin-4-yl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(4-methylbenzoyl)piperidin-4-yl]imidazolidine-2,4-dione