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N-(4-acetylphenyl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
methyl (2S,4R)-4-(2-methylquinoline-4-amido)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
2-methoxy-N-[(2R,3R)-2-methoxy-1'-(5-methylpyrazine-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
3-{[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}propan-1-ol
9-ethyl-1-methyl-4-[4-(trifluoromethyl)pyridin-2-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(1S,5R)-3-(3-chloro-4-methylbenzoyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl[3-(methylsulfanyl)propyl][(5-phenyl-1,2-oxazol-3-yl)methyl]amine
3-ethyl-N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl][(4-methoxynaphthalen-1-yl)methyl]methylamine
2-(dimethyl-1,3-thiazol-5-yl)-1-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]ethan-1-one
N5,N5-dimethyl-N6-[3-(pyridin-3-yloxy)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-[3-(4-chlorophenyl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3,3-dimethyl-1-({5-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
N-cyclopropyl-3-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]propanamide
methyl 3-[(3S,4R)-1-[(2,6-difluorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-[(5-methylhex-5-en-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)azetidin-3-yl]pyridine
5-acetyl-N-[(6-methylpyridin-2-yl)methyl]thiophene-2-carboxamide
4-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]-2-[2-(3-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
methyl 3-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]benzoate
({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-(thian-4-yl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
8-methoxy-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[2-(3,5-difluorophenyl)acetyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(2S)-N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-acetamidopropanamide
N-{2-[(3-{[(4-fluoro-3-methoxyphenyl)methyl]amino}-5-[(2-methylphenyl)sulfamoyl]phenyl)formamido]ethyl}acetamide
N-({8-[(4-ethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
N-(2-methanesulfonylethyl)-3-(2-methyl-1H-indol-1-yl)propanamide
1-(cyclohexylmethyl)-3-{2-[4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazin-1-yl]-2-oxoethyl}-3-phenylpyrrolidine-2,5-dione
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
6-chloro-2-({3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}methyl)-1,4-dihydroquinolin-4-one
ethyl 4-benzyl-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylate
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethyl-1,2-oxazole-3-carboxamide
4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-2-(trifluoromethyl)morpholine
(4aS,7aR)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(1H-imidazol-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(3-chlorophenyl)-N-(2-hydroxyethyl)-N-propylimidazo[2,1-b][1,3]thiazole-3-carboxamide
9-(2-aminopyridine-4-carbonyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclooctyl-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(benzyloxy)-8-(2,5-difluorobenzoyl)-1,8-diazaspiro[4.5]decan-2-one
1-(cyclopentylcarbamoyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
7-(3-chloro-4-hydroxybenzoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
4-[1-(2,3-dimethylbenzoyl)piperidin-3-yl]-5-(4-fluorophenyl)-2-methylpyrimidine
5-{6-chloroimidazo[1,2-a]pyridin-2-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidine
4-{[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-N-methyl-1,3-thiazol-2-amine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperazine