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[(5-ethylpyridin-2-yl)methyl](furan-2-ylmethyl)(prop-2-en-1-yl)amine
1-[(4-methanesulfonylphenyl)methyl]-2-(2-methoxyethyl)piperidine
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-[2-(2-methylphenyl)ethyl]piperidine
3-(3-fluorophenyl)-N-[2-hydroxy-2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-{3-[methyl(phenyl)amino]propyl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
3,5-dimethyl-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-1H-pyrrole-2-carboxamide
(1S,5R)-3-benzyl-6-(1-methyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,9aR)-3-ethyl-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2,5-dimethyl-3-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
1-(naphthalen-1-ylmethyl)-4-[(oxan-4-yl)amino]pyrrolidin-2-one
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
9-(3,5-dimethylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}acetamide
4-methoxy-N-[1-(1-propanoylpiperidin-4-yl)-1H-pyrazol-5-yl]benzamide
2-[(3aS,6aS)-1-(3-phenylpropyl)-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]benzonitrile
4,6-dimethyl-2-{4-[4-(piperidin-3-yl)benzoyl]piperazin-1-yl}pyrimidine
3-methoxy-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}benzamide
N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-methyl-2-(pyridin-4-yl)quinoline-4-carboxamide
6-cyclopentyl-N,1-dimethyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-5-[2-(thiophen-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,6R)-N-[(3-methylphenyl)methyl]-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5-propyl-1,3,4-oxadiazol-2-amine
6-[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
N-{3-[(4aS,8aR)-1-butyl-2-oxo-decahydro-1,6-naphthyridin-6-yl]-3-oxopropyl}methanesulfonamide
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-[(2E)-3-phenylprop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2R,3R)-2-methoxy-1'-[(4-methoxy-3-methylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
[(3R,4S)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
2-methyl-4-{4-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}butan-2-ol
1-(3-methyl-1H-indole-2-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-{5-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
(2E)-N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]-3-(thiophen-2-yl)prop-2-enamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
2-(2-oxopiperidin-1-yl)-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}acetamide
2-{[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]amino}pyridine-3-carbonitrile
(3S,4R)-1-(4-aminopyrimidin-2-yl)-3-ethyl-4-methylpiperidin-4-ol
1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(4-methylphenoxymethyl)piperidine
1-{2-oxa-7-azaspiro[4.5]decan-7-yl}-3-phenoxypropan-1-one
7-[(2,3-dimethoxyphenyl)methyl]-2-(ethanesulfonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[2-methyl-4-(1H-pyrazol-3-yl)phenoxy]acetamide
(4aR,8aS)-1-(2,3-dihydro-1H-inden-2-yl)-6-(2-fluorobenzoyl)-decahydro-1,6-naphthyridine
2-cyclobutaneamido-7-oxo-N-[2-(propan-2-yloxy)ethyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
N-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}oxan-4-amine
methyl 3-{[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}propanoate
N-[(2S,4S,6R)-2-(1,4-dimethylpiperidin-4-yl)-6-(3-hydroxyphenyl)oxan-4-yl]acetamide
(2R,4S)-4-hydroxy-1-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}piperidine-2-carboxylic acid
8-chloro-N-[(3S,5S)-1-ethyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]quinoline-2-carboxamide
2-{1-[(5-methylfuran-2-yl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
8-chloro-2-(furan-2-yl)-N-[(3R)-piperidin-3-yl]quinoline-4-carboxamide
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide