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2-{4-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}-N,N-diethylacetamide
N-[3-(4-hydroxyphenyl)propyl]-2-[methyl(piperidin-4-yl)amino]acetamide
N-({7-[4-(dimethylamino)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
N-methyl-N-(4-methylpentan-2-yl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(1R,3s,6r,8S)-4-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
1-(2-methoxy-4-methylbenzenesulfonyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine
1-(4-methoxyphenyl)-6,6-dimethyl-4-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}piperazin-2-one
2-[4-(4-fluorophenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-[4-(methylsulfanyl)phenyl]acetamide
2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-[6-(cyclopropylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,4-diazepane-1-carbaldehyde
1-[4-(4-fluorophenoxy)piperidin-1-yl]-2-(3-hydroxypiperidin-1-yl)ethan-1-one
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-1,2,3-thiadiazole-4-carboxamide
methyl 8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
3-{[(1-hydroxybutan-2-yl)[(2-methylphenyl)methyl]amino]methyl}phenol
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-(1H-1,2,4-triazol-5-yl)benzamide
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
3-(2-tert-butylphenyl)-1-{2-[(pyridin-3-yl)amino]ethyl}urea
1-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidine-1-carbonyl}pyridin-2-ol
3-({[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-6-methyl-1,2-dihydroquinolin-2-one
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]urea
4-methoxy-N-(1-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
5-(2-{2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-[2-(3-acetylpiperidin-1-yl)-2-oxoethyl]-3-(2-chlorophenyl)-1-methylpyrrolidine-2,5-dione
5-(2,3-dimethoxyphenyl)-3-(oxolan-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}azocane
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
3-[1-(4-fluoro-2-hydroxybenzoyl)piperidin-3-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
N-(2-hydroxyethyl)-5-(2-phenylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(4aS,7aR)-1-(pyridazine-3-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
2,6-dimethoxy-4-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}phenol
N-(1-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}-1-oxopentan-2-yl)acetamide
1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-4-(pyrrolidine-1-carbonyl)piperidine
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-1-methyl-1H-pyrazole-4-carboxamide
2-[2-(azepan-1-yl)acetyl]-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-methylpyridine
N-[2-(1,3-benzothiazol-2-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)benzamide
1-(oxolan-2-ylmethyl)-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperazine
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
4-[2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]piperazin-2-one
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanamide
2-(dimethylamino)-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)acetamide
4-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
3-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]azetidin-3-yl}pyridine
3-(2H-1,3-benzodioxol-5-yl)-N-[(3-methylpyridin-2-yl)methyl]-3-phenylpropanamide
(2S)-2-amino-3-hydroxy-1-[3-(3-methoxyphenoxy)azetidin-1-yl]propan-1-one
N-(2-{7-[(2E)-4-methylpent-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide