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2-(2-methoxyphenyl)-5-methyl-4-{pyrazolo[1,5-a]pyridin-7-ylmethyl}-1,3-oxazole
1-(3-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(2S)-2-(methoxymethyl)-N-[4-(1H-pyrazol-4-yl)phenyl]pyrrolidine-1-carboxamide
5-{3-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-3-oxopropyl}-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
4-(5-methylpyridin-2-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-ol
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(3-methylphenyl)methyl]pyrrolidin-2-one
5-{[1-(2-hydroxyethyl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]methyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-(2-methoxyethyl)-3-methyl-4-({[2-(3-methylthiophen-2-yl)ethyl]carbamoyl}amino)benzamide
4-(2,4-difluorophenyl)-3-(1-ethoxypropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({6-[4-(1H-imidazol-2-yl)piperidin-1-yl]pyridin-3-yl}methyl)morpholine
8-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
4-{2-[4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]ethyl}morpholine
3-acetyl-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
(3S,9aR)-8-[(3,4-difluorophenyl)methyl]-3-[(1R)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[7-(1-benzofuran-2-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
4-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-6-methoxy-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)cyclopropanamine
3-(2,5-dihydroxy-2-methylpentyl)-1-[4-(2-fluorophenoxy)phenyl]urea
methyl 9-(cyclopentyloxy)-3-[(2,6-dimethoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1R,5S)-6-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
8-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[7-(2-ethylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-3,5-dimethylbenzamide
2-(1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-2-yl)pyridine
4-[5-methyl-4-(thiophen-2-yl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-[2-(3-fluorophenyl)ethyl]-2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetamide
2-{[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline
N-[(3R,4S)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-propoxyacetamide
methyl 2-(3-acetamidophenyl)-6-methylpyridine-4-carboxylate
methyl 3-[(furan-2-ylformamido)methyl]-5-(quinoline-8-sulfonamido)benzoate
4-methyl-2-(piperidin-1-yl)-6-(pyrimidin-5-yl)pyrimidine
1-(3-{4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
2-methoxy-N-[(2R,3R)-2-methoxy-1'-(3-phenylpropanoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methyl-1H-pyrazole-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[3-(dimethylamino)pyrazin-2-yl]pyrrolidin-3-yl]-2-(propan-2-yloxy)acetamide
N-[(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]oxolane-3-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(morpholin-4-yl)-2-oxoacetamide
N-cyclopropyl-N-{[4-(methylsulfanyl)phenyl]methyl}-2-(piperidin-1-yl)acetamide
1-ethyl-3-(morpholine-4-carbonyl)-N,N-bis(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(3-methoxyphenyl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
N-[(3,5-difluorophenyl)methyl]-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
1-[(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1H-indol-3-yl)acetamide
6-[2-(hydroxymethyl)phenyl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N-cyclopropyl-2,6-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]quinoline-4-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
4-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}piperazine-1-carboxamide
N-methyl-3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
6-(naphthalene-1-carbonyl)-N-[3-(2-oxoimidazolidin-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
7-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-2,7-diazaspiro[4.4]nonane-1,3-dione