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2-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-4,6-dimethylpyridine-3-carbonitrile
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1,3-thiazole-4-carboxamide
1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
methyl (2S,4S)-1-[(2-chlorophenyl)methyl]-4-acetamidopyrrolidine-2-carboxylate
4-methyl-7-[2-(1-methylpiperidin-4-yl)-1H-imidazol-1-yl]-2H-chromen-2-one
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
2-methyl-4-[5-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)thiophen-2-yl]but-3-yn-2-ol
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
2-(4-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-ol
1-(furan-2-ylmethyl)-N-[2-(1,3-thiazol-2-yl)ethyl]piperidine-3-carboxamide
N-(2,6-dimethylphenyl)-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
{[6-(pyrrolidin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}({[2-(trifluoromethyl)phenyl]methyl})amine
2-(2-methoxyphenyl)-8-methyl-5-[(4-methyl-1H-imidazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-({5-[1-(4-methoxypyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
N-(2-{4-[(3-hydroxyphenyl)methyl]morpholin-2-yl}ethyl)-1,2,5-oxadiazole-3-carboxamide
{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
N-[2-(1H-indol-1-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-cyclohexyl-N-[3-(dimethylamino)-2,2-dimethylpropyl]-1H-pyrazole-4-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-[(1S,5R)-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-cyclopropyl-1-[2-(4-fluoro-2-methylphenyl)acetyl]piperazine-2-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
4-(2-hydroxy-5-methylbenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
1-(2-fluorophenyl)-4-({4-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)piperazine
4-methoxy-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)benzamide
N-[2-(3-acetamidophenyl)phenyl]butanamide
4-[2-(azetidine-1-carbonyl)-4-methoxyphenoxy]-1-cyclopropanecarbonylpiperidine
N-(oxolan-2-ylmethyl)-3-phenyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(pentan-3-yl)carbamoyl]pyrrolidine-2-carboxylic acid
3-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidine-1-carbonyl]-1,5,6-trimethyl-1,2-dihydropyridin-2-one
1-({3-[3-(diethylamino)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)azetidin-3-ol
4-(hydroxymethyl)-1-(1H-indol-7-ylmethyl)azepan-4-ol
N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-1-methylpyrrolidine-3-carboxamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-[(3-methoxypiperidin-1-yl)sulfonyl]-N-(1,2-oxazol-3-ylmethyl)benzamide
1-(3-{[4-(hydroxymethyl)-4-[(4-methoxyphenyl)methyl]piperidin-1-yl]methyl}phenyl)ethan-1-one
3-{1-[(6-ethoxypyridin-3-yl)methyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-chloro-5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(2-fluorophenyl)-N-[2-(1H-imidazol-4-yl)ethyl]cyclopropane-1-carboxamide
5-[4-({2-[(4-methoxyphenyl)amino]-1,3-thiazol-5-yl}methyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
1-[3-(2-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}-4-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-3-yl)morpholine
5-(3-methoxyphenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1,2,4-triazin-3-amine
1-[2-(2-chlorophenyl)-2-hydroxyacetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]-2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}acetamide
4-ethyl-6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-(pyrrolidin-1-yl)pyrimidine
{1-[3-(4H-1,2,4-triazol-4-yl)propyl]piperidin-3-yl}methanol
N-{3-[ethyl(methyl)amino]butyl}-6-(propan-2-yl)pyrimidin-4-amine
3-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
2-ethyl-5-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,3,4-oxadiazole