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4-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
4-[(2H-1,3-benzodioxol-4-ylmethyl)amino]-1-(3-phenylpropyl)pyrrolidin-2-one
N-({8-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)cyclohexanecarboxamide
1,3-dimethyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-1H-pyrazole-5-carboxamide
N-(2,3-dihydroxypropyl)-N,5-dimethyl-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]propanamide
N-[2-(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclohexanecarboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-6-(piperidin-3-yl)pyrimidin-4-amine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
8-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-(1H-indol-1-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-methyl-3-{[methyl({[1-(2-methylphenyl)-1H-1,2,3,4-tetrazol-5-yl](phenyl)methyl})amino]methyl}pyridin-2-amine
2,4-dimethyl-N-[4-(4-{[1-(thiophen-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]benzamide
N-(propan-2-yl)-1-[(1s,4s)-4-(quinoline-8-sulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-methoxy-3-{[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
1-[1-(4-ethylbenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
N-(1-{7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
2-[({5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)sulfanyl]pyrimidine
N-[2-(2-fluorophenoxy)ethyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
N-[2-(2,4-difluorophenyl)-1-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}ethyl]-N-methylpyridine-3-carboxamide
4-(3-methoxypyrazin-2-yl)-1-phenylpiperazin-2-one
(2S,4R)-N-(1-benzothiophen-2-ylmethyl)-1-(cyclohexylmethyl)-N-methyl-4-[(4-methylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
8-cyclopropanecarbonyl-2-[(2-fluoro-3-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
3-{[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]sulfonyl}-N-methylbenzamide
1-{3-[4-(benzyloxy)piperidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
N-[2-(4-hydroxyphenyl)ethyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
5-[4-(thiomorpholin-4-yl)piperidin-1-yl]pentan-1-ol
11-(4-ethylpiperazin-1-yl)-4-[(4-fluorophenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
ethyl 1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-(3-hydroxy-3-phenylpropyl)-5-methoxy-N,1,2-trimethyl-1H-indole-3-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(3-methoxyphenyl)ethyl]benzamide
2-{[3-(pyridin-4-yl)azetidin-1-yl]methyl}benzonitrile
N-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
3-{4-[5-(2-methoxybenzamido)-1H-pyrazol-1-yl]piperidin-1-yl}propanoic acid
methyl 3-(4-{[(5-oxo-1-phenylpyrrolidin-3-yl)amino]methyl}-1H-pyrazol-1-yl)propanoate
4-[2-(pyrrolidine-1-carbonyl)phenoxy]-1-{[2-(trifluoromethyl)phenyl]methyl}piperidine
4-{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-indole-5-carboxamide
(4S)-1-[(2-fluoro-4-methoxyphenyl)methyl]-3,3,4-trimethylpiperidin-4-ol
(4S,4aS,8aS)-4-phenyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-decahydroquinolin-4-ol
2-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-(3-methylpiperidin-1-yl)ethan-1-one
2-amino-7-methyl-4-[3-(pyridin-2-ylmethoxy)phenyl]-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
4-{1-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]ethyl}morpholine
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[4-(trifluoromethyl)benzoyl]piperidine
2-[2-(dimethylamino)pyrimidin-5-yl]-N,N-dimethylquinoline-4-carboxamide
N-[3-(2-chlorophenoxy)propyl]-5-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(2H-1,3-benzodioxol-5-yl)-5-(1H-pyrazol-3-yl)-1H-1,2,4-triazole