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5-cyclopropanecarbonyl-1'-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(4-fluoro-3-methoxyphenyl)methyl](methyl)(oxan-4-ylmethyl)amine
(3S,4R)-1-(2,3-dimethyl-1H-indole-7-carbonyl)-4-methylpiperidine-3,4-diol
(2S)-2-amino-3-(1H-indol-3-yl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]propanamide
5-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
1-[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-[(5-chlorothiophen-2-yl)methyl]-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
2-ethyl-8-(5-methyl-2-phenylfuran-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S)-1-(3-fluoropyridine-4-carbonyl)-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2,6-difluorobenzamide
1-(2-phenylpropyl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
(2S,4R)-N,1-dimethyl-4-[4-(5-methylfuran-2-yl)benzamido]pyrrolidine-2-carboxamide
2-(cyclohexylmethyl)-4-(1-methyl-1H-pyrazole-5-carbonyl)morpholine
3-[3-(3-methylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl]piperidine-1-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2,3-dihydro-1-benzofuran-7-carboxamide
(2S,4R)-1-[(3-fluorophenyl)methyl]-N-methyl-4-[(5-propyl-1,3,4-thiadiazol-2-yl)amino]pyrrolidine-2-carboxamide
1-(4-methylpiperidin-1-yl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propan-1-one
N-(2-methanesulfonamidoethyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-(2-fluorophenyl)cyclopropane-1-carboxamide
N-({7-[2-(2,6-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)pyrazine-2-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-(1H-pyrazol-1-yl)benzamide
2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyridin-2-yl)phenol
2-(6-aminopyridin-3-yl)-2-{methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetic acid
N-(1-hydroxybutan-2-yl)-N-[(5-methylthiophen-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
(3S,4R)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
(1S,5R)-6-(2-ethylpyrimidine-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(1H-indol-3-yl)ethyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl[(3-{[1-(4-methylbenzoyl)piperidin-4-yl]oxy}phenyl)methyl][2-(1H-1,2,4-triazol-1-yl)ethyl]amine
3-{[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]sulfamoyl}-N-(prop-2-en-1-yl)benzamide
9-ethyl-1-methyl-4-[2-(pyridin-3-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(2E)-N-{[3-methyl-7-(naphthalene-1-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
4-(3-chlorothiophene-2-carbonyl)-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[3-(2-{[(3,4-difluorophenyl)methyl]carbamoyl}ethyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
3-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)-N-(trimethyl-1H-pyrazol-4-yl)benzamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2-dimethyl-2-(morpholin-4-yl)propanamide
methyl N-(2-oxo-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)carbamate
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(2-fluoro-4-methoxyphenyl)methyl]amine
5-(2-fluorophenyl)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
6-{4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}pyridine-2-carboxylic acid
5-{3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-3-oxopropyl}-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
2-ethyl-4-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1-methylpiperazine
[(3R,4R)-1-[2-(difluoromethoxy)benzoyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
8-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-2-benzyl-2,8-diazaspiro[4.5]decan-3-one
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-[(1-hydroxycyclohexyl)methyl]propanamide
5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-(cyclopropylmethyl)-5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide