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4-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-4-yl]pyridine
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-5-methoxy-1-methyl-1H-indole
1-(cyclohexylmethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-6-oxopiperidine-3-carboxamide
5-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]thiophene-2-carboxylic acid
N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]-2-hydroxyacetamide
N-benzyl-N-(2-phenylethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
5-(2-phenylethyl)-5-[1-(pyridin-4-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
1-(2-methoxyacetyl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-3-carboxamide
6-{[methyl(2-phenylethyl)amino]methyl}-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide
[5-methyl-7-(1-methyl-1H-1,2,3,4-tetrazol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
3-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
5-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
ethyl 4-{6-[(3-phenoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-amido}piperidine-1-carboxylate
N-[2-(dimethylamino)ethyl]-N-(2-hydroxyethyl)-2-methyl-1-benzofuran-7-carboxamide
2-[3-(azepane-1-carbonyl)piperidin-1-yl]-7-methanesulfonyl-4-methylquinazoline
3-(pentan-2-yl)-8-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4R)-3-methoxy-1-(2,3,4-trimethoxybenzoyl)piperidin-4-amine
4-[(2S,4R)-1-[(2-ethoxyphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
1-(cyclopropylmethyl)-5-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]naphthalene-2-carboxamide
2-(2-phenylethyl)-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[1-(3-chlorobenzoyl)piperidin-4-yl]-5-phenyl-2-(pyridin-3-yl)pyrimidine
6-[5-chloro-2-(propan-2-yloxy)phenyl]pyrimidin-4-amine
N-cyclobutyl-5-(2,6-dimethoxyphenyl)-1,2,4-triazin-3-amine
N-[2-(2-fluorophenyl)-1-[1-(oxolane-3-carbonyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
2-methyl-6-{[4-(4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidin-1-yl)piperidin-1-yl]methyl}pyridine
[(3-{[1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-3-ylmethyl)amine
1,3,7-trimethyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1H-indole-2-carboxamide
2-(3-hydroxyphenyl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N,5-dimethyl-1-propyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(2-hydroxypropyl)-9-(1H-imidazol-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2,4-dimethoxy-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]benzamide
6-[(4-hydroxy-3-methoxyphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-6-azaspiro[2.5]octane-1-carboxamide
1-benzyl-4-oxo-N3-[(4-phenyloxan-4-yl)methyl]-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
5-[1-(3-chlorothiophene-2-carbonyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-[4-(2,3-dimethoxyphenyl)phenyl]-2-methylpropanamide
N,N,7-trimethyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
N-methyl-3-[methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amino]butanamide
N-(2-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
(2E)-N-[2-(8-methoxyquinolin-5-yl)phenyl]but-2-enamide
N-benzyl-1-methyl-N-[(1R,3S,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-({7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)oxolane-3-carboxamide
2-(cyclohex-1-en-1-yl)-N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N3-(furan-2-ylmethyl)-N5-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,1-dimethylpiperidine-2-carboxamide
methyl({[1-(2-methylpropyl)pyrrolidin-3-yl]methyl})[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-(2-{7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
2-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-4,6-dimethylpyridine-3-carbonitrile
(oxan-2-ylmethyl)({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine