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2-(4-{[2-(2-chloro-6-methylphenoxy)ethyl]amino}cyclohexyl)acetic acid
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-3-methylthiophene-2-carboxamide
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]phenoxy}acetamide
1-(1,3-benzothiazol-2-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}piperidin-4-amine
5-(azocane-1-carbonyl)-1-(2-ethoxyethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
[1-(2-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}ethyl)piperidin-2-yl]methanol
N-(2-{7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
1-(3-methoxypropyl)-8-[(5-methylthiophen-2-yl)methyl]-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(dimethyl-1,2-oxazol-4-yl)-N-[3-(2,6-dimethylphenoxy)propyl]-N-methylpropanamide
N-(2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)acetamide
5-chloro-6-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]pyridine-3-carboxylic acid
3-(2,4-dimethoxyphenyl)-1-[(1-methylpiperidin-4-yl)methyl]urea
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
8-(2-amino-2-methylpropyl)-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3-{2-[1-(5-chlorothiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyridine-2-carbonitrile
2-methyl-5-(3-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1,3,4-thiadiazole
2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]-4-phenylphenol
3-(4-benzylpiperazine-1-carbonyl)-2-(cyclopentylmethyl)-1-(3-methoxypropyl)-6-methyl-1,4-dihydropyridin-4-one
methyl 2-(2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
2-methyl-6-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
N,N-diethyl-2-(4-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-1H-1,2,3-triazol-1-yl)acetamide
methyl (2S)-3-phenyl-2-{[1-(3-phenylpropyl)-1H-1,2,3-triazol-4-yl]formamido}propanoate
(3aS,6aS)-2-(dimethylsulfamoyl)-5-(6-methylpyridazin-3-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}benzoic acid
4-{[(2H-1,3-benzodioxol-5-ylmethyl)(methyl)amino]methyl}-N-(1-methyl-1H-pyrazol-4-yl)benzamide
3-(3-fluorophenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1H-pyrazole-4-carboxamide
3-ethyl-1-methyl-N-({3-methyl-7-[2-(thiophen-2-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-pyrazole-5-carboxamide
methyl 4-(5-chloro-2-{[2-(pyridin-4-ylsulfanyl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
3-(1H-imidazol-2-yl)-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[cyclohexyl(methyl)amino]-3-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenoxy)propan-2-ol
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(2-oxoazonan-1-yl)acetamide
4-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-6-(morpholin-4-yl)pyrimidin-2-amine
methyl 1-ethyl-5-{[(4-methoxy-3-methylphenyl)methyl]amino}-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl 5-{[4-(difluoromethoxy)phenyl]methyl}-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(3-fluorophenyl)propanamide
2-cyclopropyl-9-(2,3-dihydroxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(2E)-1-[(4aR,8aS)-6-cyclopropanecarbonyl-decahydro-1,6-naphthyridin-1-yl]-2-methylbut-2-en-1-one
2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
[2-(isoquinolin-5-yl)phenyl]methanol
N-cyclopropyl-1-(2-{1-[(2,4-dimethoxy-3-methylphenyl)methyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
ethyl 4-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}piperazine-1-carboxylate
N-cyclopropyl-5-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-(oxolan-3-yl)-5-[4-(propan-2-yl)phenyl]-1,2,4-oxadiazole
(1r,4r)-4-({[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)cyclohexane-1-carboxamide
[3-(1H-1,2,3-benzotriazol-1-yl)propyl]({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl})amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[5-(morpholin-4-yl)pentyl]benzamide
[(3R,4R)-1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-[2-(azepan-1-yl)-2-oxoethyl]-3-(2-chlorophenyl)-1-cyclopentylpyrrolidine-2,5-dione
2-{[2-(propan-2-ylsulfanyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid