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N4-[1-(2,6-dimethylphenoxy)propan-2-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}benzamide
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-[(1-phenylcyclohexyl)methyl]acetamide
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
4-(oxane-4-carbonyl)-7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 5-[(2,5-dimethoxyphenyl)methyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
methyl 2-(3-{[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]methyl}-1H-indol-1-yl)acetate
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
(2S,4R)-4-butanamido-N,N-diethyl-1-[(trimethyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
N-methyl-2-(morpholin-4-yl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-3-yl)acetamide
4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
1-tert-butyl-N-{2-[methyl(phenyl)amino]ethyl}-5-oxopyrrolidine-3-carboxamide
6-{1-[(2E)-5-methyl-2-(propan-2-yl)hex-2-en-1-yl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
methyl (2S,4R)-4-(2-methylpropanamido)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
N-{[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropanecarboxamide
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]propanamide
N-[2-(2,4-dimethylphenoxy)ethyl]-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-cyclopropyl-N-[2-(1H-indol-3-yl)ethyl]-N-(pyridin-3-ylmethyl)-1H-pyrrole-2-carboxamide
5-[(3-methoxyphenyl)methyl]-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-phenoxy-N-(1-{7-[(2,3,4-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
2-(3,5-dimethoxyphenyl)-1-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
ethyl({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})[(4-phenyl-1,3-thiazol-2-yl)methyl]amine
N3-(1-benzylpyrrolidin-3-yl)-N5-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]benzamide
6-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-3,5-dimethoxy-N-[(4-methoxyphenyl)methyl]benzamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperidine
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]pyrrolidine-3-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
6-(quinolin-3-yl)pyridine-3-carboxamide
1-methyl-4-{[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
5-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N2-(3-methylphenyl)-6-{2-oxa-7-azaspiro[4.5]decan-7-ylmethyl}-1,3,5-triazine-2,4-diamine
N-benzyl-2-(4-{4-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}phenyl)acetamide
6-tert-butyl-N-(1,4-dioxan-2-ylmethyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{4-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-4-oxobutyl}piperidin-2-one
(2,1,3-benzoxadiazol-5-ylmethyl)({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl})amine
1-[(4aR,8aS)-6-[2-(thiophen-2-yl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-2-(4-chloro-2-methylphenoxy)propan-1-one
3-(2-chlorophenyl)-6-(pent-4-enoyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
[(3R,4R)-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
2,4-dimethyl-N-[4-(4-{[1-(pyridin-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]benzamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-3-(2-oxoazepan-1-yl)propanamide
1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(pyridin-2-yl)propan-1-one
2-{2-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}pyrazine
[3-(hydroxymethyl)-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl]methanol
5-(1-cycloheptyl-1H-1,2,3-triazol-4-yl)-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
ethyl 4-benzyl-1-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]piperidine-4-carboxylate