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1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-(piperidine-1-carbonyl)piperidine
5-{1-[2-(4-chlorophenyl)acetyl]piperidin-4-yl}-3-(2,3-dihydro-1H-inden-2-yl)-5-methylimidazolidine-2,4-dione
N-[2-(diethylamino)ethyl]-N-methyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(3-chloro-4-hydroxyphenyl)-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}acetamide
3-[({[4-(2-methoxyethoxy)phenyl]methyl}carbamoyl)amino]-N,N-dimethylbenzamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
4-hydroxy-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
methyl 5-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-3-acetamido-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-acetyl-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)piperidine-4-carboxamide
ethyl 1-[(4-fluorophenyl)carbamoyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
methyl 1-(2-methoxyethoxy)-2-oxo-8-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
(3R,4R)-1-[4-(3-chlorophenyl)pyrimidin-2-yl]-4-ethylpiperidine-3,4-diol
8-(1-aminocyclopropanecarbonyl)-3-[2-(4-ethylpiperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-{[4-(2-aminoethyl)phenyl]methyl}-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(2-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
4-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-6-methyl-1,2-dihydroquinolin-2-one
4-{3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}-4H-1,2,4-triazole
2-(3-fluorophenyl)-N-{[7-(2-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
4-methyl-5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-imidazole
(1S,5R)-6-(dimethyl-1,2-oxazole-4-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
4-(4-fluorophenyl)-2-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenol
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]acetamide
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-[4-(2,6-dimethylquinoline-3-carbonyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
2-{4-[(2-chlorophenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
2-(4-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
methyl 1-(3-{3-[(cyclohexylamino)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
2-ethyl-N-(1H-indol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-[4-(cyclopropylmethoxy)phenyl]-2-[4-(pyridin-4-yl)piperidin-1-yl]acetic acid
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-(3-acetylphenyl)-3-(2-aminoethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-(4-{1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}phenyl)ethane-1-sulfonamide
N-{[6-chloro-4-(cyclopentylamino)quinazolin-2-yl]methyl}-2-ethylbutanamide
[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]({[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl})amine
1-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-cyclopentyl-4-methyl-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)benzamide
2-[4-(3,3,5,5-tetramethylcyclohexyl)piperazin-1-yl]pyridine-4-carboxamide
3-methyl-1-{1-[6-(piperazin-1-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](methyl)(pyrazin-2-ylmethyl)amine
1-{3-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
3-{1-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]azetidin-3-yl}pyridine
N3-[(4-fluorophenyl)methyl]-N5-[1-(furan-2-yl)ethyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[(1S,5R)-6-(2-propoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
15-methyl-12-(4-propylpiperazine-1-carbonyl)-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
3-methyl-N-{[8-(pyridin-3-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}pentanamide
6-(4-methoxyphenyl)-N-(2-methylpropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide