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2-{4-[3-(2,3-dimethoxyphenyl)pyrrolidine-1-carbonyl]piperidin-1-yl}-6-fluoro-4-methylquinazoline
2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-6-methylpyridine-3-carbonitrile
methyl 2-{[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl](methyl)amino}acetate
N-(1H-indol-2-ylmethyl)-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
6-(2-chlorophenyl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[(cyclohex-1-en-1-ylmethyl)amino]-N-[(2-methoxyphenyl)methyl]acetamide
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
(1R,3S)-3-(2-hydroxyethoxy)-7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-7-azaspiro[3.5]nonan-1-ol
methyl 4-(3-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propanamido)benzoate
N-{[2-(2-methylpyridin-4-yl)phenyl]methyl}propanamide
N-[(3,4-difluorophenyl)methyl]-2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-{2-oxo-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-(thiophen-2-ylmethyl)acetamide
6-chloro-N,N-dimethyl-3-({[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
4-[1-(2H-1,3-benzodioxol-5-yl)-3-(pyridin-3-yl)prop-2-yn-1-yl]morpholine
propyl (4aR,7aS)-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
N-[2-(3-methoxyphenyl)-1-{1-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carbonyl]piperidin-4-yl}ethyl]-N,3-dimethylbutanamide
4-chloro-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
3,5-dimethoxy-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
1-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(propan-2-yl)urea
(1S,5R)-3-[2-(2,3-dimethylphenoxy)ethyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(3-methoxypropyl)acetamide
2-acetyl-8-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[(3-chloropyridin-4-yl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazine
6-{3-[(4-fluorophenyl)amino]piperidine-1-carbonyl}-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
N-butyl-N-methyl-3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-[(2R,3R)-1'-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
1-(4-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}thiophen-2-yl)ethan-1-one
ethyl 1-[3-(methylsulfanyl)propanoyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
4-(2,2-diphenylethyl)-3-[2-oxo-2-(3-oxopiperazin-1-yl)ethyl]piperazin-2-one
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-(2-oxopyrrolidin-1-yl)benzamide
(2S,4R)-4-amino-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(butan-2-yl)-N-[(4-methylphenyl)methyl]-3-(1-methylpiperidin-4-yl)propanamide
2-{4-[2-(1H-imidazol-2-yl)benzoyl]piperazin-1-yl}-4,6-dimethylpyrimidine
{5-[1-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]furan-2-yl}methanol
N'-[(5-chloro-2-methoxyphenyl)methyl]-N-cyclopentyl-N'-methylbutanediamide
(4aS,8aR)-6-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-cyclopentyl-2-{[(4-methyl-2-phenyl-1,3-thiazol-5-yl)methyl]amino}propanamide
5-[(3-fluorophenyl)methyl]-5-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-3-(2-methylpropyl)imidazolidine-2,4-dione
N-({5-methyl-2-[3-(oxane-4-amido)phenyl]-1,3-oxazol-4-yl}methyl)-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
5-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-(4-{1-[(4-fluorophenyl)methyl]-1H-imidazol-2-yl}phenyl)-2-methylbut-3-yn-2-ol
2-[(1S,5R)-6-[(2,5-difluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
2-[4-(4-methyl-1H-imidazole-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
4-ethenyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}benzamide
3-{1-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-3-yl}benzoic acid