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N-cyclopropyl-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-[(5-methylthiophen-2-yl)methyl]propanamide
5-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
1-[(4aS,8aR)-decahydroisoquinolin-2-yl]-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-3-(pyridin-3-yl)propan-1-one
2-(2-chlorophenyl)-2-hydroxy-1-{4-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}ethan-1-one
2-(4-chlorophenoxy)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
4-[(3-ethenylphenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-(2-acetylphenyl)-5-(azepane-1-sulfonyl)benzoic acid
N-[3-(4-{[2-(2H-1,3-benzodioxol-5-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-1-methylpiperidine-3-carboxamide
2-{1-[(4-methylphenyl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2,3,4-trimethoxy-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
N-[2-(dimethylsulfamoyl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(3S,4R)-1-[(3-chloro-4-fluorophenyl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
6-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-sulfonyl}-1,2,3,4-tetrahydroquinolin-2-one
[(3-chloro-4,5-diethoxyphenyl)methyl][1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(2-hydroxyethyl)amino]pyridine-3-carboxamide
1-[(4-methyl-1,3-thiazol-5-yl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
8-cyclobutyl-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
3-[2-(4-benzylpiperazin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
7-(4-chloro-1H-indole-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[4-(benzenesulfonyl)piperazin-1-yl]-3-(pyridin-2-yl)propan-1-one
ethyl 4-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]piperidine-1-carboxylate
1-[(4-chlorophenyl)methyl]-4-[(2,3-difluoro-4-methoxyphenyl)methyl]piperazine
methyl 2-[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-6-methylpyrimidine-4-carboxylate
(1S,2S)-N2-[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]-2,3-dihydro-1H-indene-1,2-diamine
N-[2-(4-fluorophenyl)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-ethyl-3-[2-oxo-2-(5-oxo-1,4-diazepan-1-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
1-(carbamoylmethyl)-N-{2-[ethyl(3-methylphenyl)amino]ethyl}piperidine-3-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
N-cyclopentyl-2-{methyl[(2E)-3-phenylprop-2-en-1-yl]amino}propanamide
5-methyl-1-[2-oxo-2-(2-phenylazetidin-1-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(3-fluorophenyl)amino]-N-(prop-2-en-1-yl)piperidine-1-carboxamide
2-[5-({2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazol-3-yl]pyrimidine
1-benzyl-8-[(3,4-dimethoxyphenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-acetamido-1-ethyl-2-(2-fluorophenyl)-N-methyl-N-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-methyl-N-phenylpiperidine-1-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylacetamide
1-(2-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-3,3-dimethylurea
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-methylpentane-1,2-dione
{3-propyl-1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl}methanol
3-[(3,4-dimethoxyphenyl)methyl]-1-ethyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-1,2,4-triazole
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(methylsulfanyl)propan-1-one
N,8-dimethyl-3-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
2-{[2-(morpholin-4-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-(3-chlorothiophene-2-carbonyl)-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{5-[(1S)-1-acetamido-3-methylbutyl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1-oxaspiro[4.4]nonan-2-one