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1-[2-(3-methylbutyl)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-en-8-yl]pentane-1,4-dione
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[3-(pyridin-2-yl)propanoyl]pyrrolidine-3-carboxylic acid
2-methyl-6-[2-(2-phenylethyl)piperidine-1-carbonyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-(3-cyclopentylpropyl)-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-methyl-4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-methyl-1,3-thiazole-4-carboxamide
2-(4-{[3-(cyclopentyloxy)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
5-fluoro-1,3-dimethyl-2-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-indole
3-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
6-fluoro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-ethyl-2-[4-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperazin-1-yl]acetamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]pyridine-3-carboxamide
methyl 5-[(2R)-2-amino-3-(1H-indol-3-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-cyclopropyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)acetamide
4-methyl-2-({methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)phenol
(3R,4R)-4-ethyl-1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]piperidine-3,4-diol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-15-methyl-9-(5-methylthiophen-2-yl)-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl]methanol
6-[(2E)-3-(1H-imidazol-4-yl)prop-2-enoyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(2-methoxyethyl)-4-(4-phenyl-5-propyl-1H-imidazol-2-yl)pyrrolidin-2-one
5-chloro-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
4-({4-benzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1-(prop-2-en-1-yl)-1H-pyrazole
{1-methyl-5-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
8-methoxy-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(3,5-dimethoxyphenyl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-(1-methyl-5-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}-1H-1,3-benzodiazol-2-yl)ethan-1-ol
methyl[(4-methyl-1H-imidazol-5-yl)methyl][2-(4-methylphenoxy)ethyl]amine
1-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)-4-(oxolane-2-carbonyl)piperazine
5-ethyl-2-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-(9H-fluoren-2-ylmethyl)-N-(furan-2-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-amino-1-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-2-methylpropan-1-one
3-(2-methoxyphenyl)-N-{1-[({[4-(1H-pyrazol-1-yl)phenyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}propanamide
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4-cyclopentylpyrimidin-2-yl)-N-[(3-methylpyridin-4-yl)methyl]piperidin-4-amine
1-propyl-4-({5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,1-dimethyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
9-[4-(dimethylamino)benzoyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[2-(piperidin-1-yl)ethyl]-7-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
6-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
3-(3-methoxyphenoxy)-1-(thiophen-3-ylmethyl)azetidine
1-(4-methanesulfonyl-1,4-diazepan-1-yl)-3-(pyridin-4-yl)propan-1-one
1-(1H-imidazol-2-ylmethyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-amino-N-(butan-2-yl)-N-[(2-chlorophenyl)methyl]-6-methylpyrimidine-4-carboxamide
2-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]quinoline
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1H-1,2,4-triazole-5-carboxamide
1-(2-methylphenyl)-4-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1,4-diazepane
N-(2,3-dihydro-1H-inden-2-yl)-2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]acetamide
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)(thiophen-3-ylmethyl)amine