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N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3R,4R)-3,4-dimethyl-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-ol
[(2-methoxynaphthalen-1-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
4-[1-(hydroxymethyl)cyclopropanecarbonyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 1-(1,4-dithiepan-6-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-(1-cyclopentanecarbonylpiperidin-4-yl)-N-cyclopropylpiperidine-3-carboxamide
2-({[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(ethyl)amino)ethan-1-ol
3-chloro-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]thiophene-2-carboxamide
(3R,4R)-4-(hydroxymethyl)-1-[4-(2-methoxyphenyl)benzoyl]piperidin-3-ol
2-methoxy-4-[(1E)-3-[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]prop-1-en-1-yl]phenol
N-[2-(dimethylamino)ethyl]-N-ethyl-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)benzoic acid
N-[1-(1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
(3R,5S)-N-butyl-5-(3-fluorophenoxymethyl)piperidine-3-carboxamide
(2R,3R)-3-amino-1'-[5-(propan-2-yl)thiophene-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(2-acetyl-4,5-dimethoxyphenyl)-1-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]ethan-1-one
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(4-methylphenyl)acetamide
1-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-methoxypropan-1-one
2-{2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-(4-fluorophenyl)-4-[4-(morpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3-acetamido-N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}benzamide
4-(2-methoxyphenoxy)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine
1-methyl-N-[2-(morpholin-4-yl)ethyl]-5-[2-(4-phenylphenyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-(benzyloxy)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]ethan-1-one
N-(4-chloro-2-fluorophenyl)-2-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)acetamide
N-methyl-3-phenoxy-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
1-ethyl-8-[(3-methylthiophen-2-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-({[3-(3-fluorophenyl)oxolan-3-yl]methyl}amino)piperidine-1-carboxylate
2-benzyl-8-[2-(2-methylphenoxy)acetyl]-2,8-diazaspiro[4.5]decan-3-one
3-{1-[5-(1-benzofuran-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-5-methyl-4H-1,2,4-triazole
3-{[3-(piperidin-1-ylmethyl)piperidin-1-yl]methyl}pyridin-2-amine
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
3,5-dimethoxy-2-{[3-(methylcarbamoyl)pyrrolidin-1-yl]methyl}benzoic acid
1-[4-(3,3-dimethyl-4-phenylpyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
2-[(dimethylamino)methyl]-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1,3-thiazole-4-carboxamide
N,N-diethyl-1-({1-[3-(3-methoxyphenyl)propanoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
3-{[4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-indole
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-2-(2-methylphenoxy)ethan-1-one
N-propyl-N-(pyridin-3-ylmethyl)-2-(thiophen-3-yl)acetamide
5-phenyl-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1,2,4-triazin-3-amine
3-(hydroxymethyl)-1-(1H-pyrazole-3-carbonyl)piperidin-3-ol
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
7-fluoro-2-methyl-4-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]quinoline
1-(2-{1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)piperidin-2-one
N-[(5-chloro-2-ethoxyphenyl)methyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
8-methyl-2-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
4-({2-[1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine