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N-[(5-chlorothiophen-2-yl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
1-cyclopropyl-5-oxo-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}pyrrolidine-3-carboxamide
[(2S)-1-(5-methyl-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-2-yl]methanol
2-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methylpyrazine
2-butyl-5-chloro-4-[1-(1-methoxypropan-2-yl)-1H-imidazol-2-yl]-1H-imidazole
N-ethyl-N-methyl-6-[methyl({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amino]pyridine-3-carboxamide
2,3-dimethyl-7-[1-(prop-2-en-1-yl)pyrrolidine-2-carbonyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-(pyrrolidin-1-yl)propan-2-ol
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
1-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]methyl}piperidine-4-carboxamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
2-methyl-1-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,4-dihydroquinolin-4-one
(3S,4R)-3-benzyl-1-(2-methoxypyridine-4-carbonyl)-4-methylpiperidin-4-ol
1-{2-oxo-2-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}pyrrolidin-2-one
7-propyl-2-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[4-(hydroxymethyl)-1,3-thiazol-2-yl]piperidin-3-ol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-ethoxy-4-(prop-2-en-1-yloxy)benzamide
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-[ethyl(methyl)amino]propan-1-one
2-[(4aS,8aR)-1-[2-(methylamino)ethyl]-2-oxo-decahydro-1,6-naphthyridin-6-yl]-N,N-dimethylpyridine-3-carboxamide
(1R,4S)-2-[2-(2-fluoro-5-methoxyphenyl)pyridine-3-carbonyl]-2-azabicyclo[2.2.1]heptane
N-{2-[(1R,7S)-6-(4-methylpiperidine-1-carbonyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-3-yl]ethyl}acetamide
8-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-1-oxa-8-azaspiro[4.5]decane
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[2-(furan-2-yl)azepane-1-carbonyl]-5-methoxy-4H-pyran-4-one
3-({2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]acetamido}methyl)-4-methylbenzoic acid
2-(5-acetylthiophen-3-yl)-1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
8-[2-(methylamino)acetyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-{2-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
5-[4-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
2-methyl-6-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylthiophene-3-carboxamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-(3-propyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
1-(3-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
2-{1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}benzoic acid
3-[1-(1H-1,3-benzodiazol-2-yl)-3-(methylsulfanyl)propyl]-1-(1,5-dimethyl-1H-pyrazol-4-yl)urea
1-(3-methoxybenzoyl)-4-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]piperidine
3-ethyl-6-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-3H-imidazo[4,5-b]pyridin-2-amine
2-[5-(2,6-dichlorophenoxymethyl)-1,2,4-oxadiazol-3-yl]pyridine
3-(3-hydroxy-3-methylbutyl)-N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]benzamide
N-[4-chloro-2-(3,4,5-trimethoxyphenyl)phenyl]acetamide
6-[4-(3-methylphenoxy)piperidine-1-carbonyl]quinoxaline
(1R,5R)-3-(4-fluorobenzenesulfonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3-methyl-N-(1-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
2-({6-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}dimethylamine
1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
8-acetyl-2-(2-methyl-2-phenylpropanoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(2-hydroxyethyl)-N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
methyl 4-({[(3S,5S)-1-[(3-chlorophenyl)methyl]-5-{[2-(2-fluorophenyl)ethyl]carbamoyl}pyrrolidin-3-yl]amino}methyl)benzoate
1-cyclobutanecarbonyl-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]piperidine-4-carboxamide