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2-methoxy-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(3aR,6aR)-2-methyl-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
1-[(2-chlorophenyl)methyl]-7-fluoro-3-({[3-(morpholin-4-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[1-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
2-(4-fluorophenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
2-(4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-2-methyl-4-phenyl-1,3-thiazole
5-methanesulfonyl-1'-(3-methoxypyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(cyclopropylmethyl)-3-hydroxy-3-[({[3-(trifluoromethyl)phenyl]methyl}amino)methyl]piperidin-2-one
2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
[1-(2-aminopyrimidin-4-yl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
6,7-dimethoxy-2-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}-4-(pyrrolidin-1-yl)quinazoline
1-[2-(1,3-dihydro-2-benzofuran-5-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(1,4-dioxan-2-ylmethyl)-N-methylpiperidine-3-carboxamide
N-[2-(4-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-4-(2-oxopyrrolidin-1-yl)butanamide
1-[2-(1H-imidazol-4-yl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-N-(propan-2-yl)pyridine-2-carboxamide
9-methoxy-10-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
({5-[1-(5-chloro-2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)dimethylamine
2-{5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl}-6-methylpyridine
methyl 4-(5-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)acetamide
1-[2-(2-methoxy-4-methylphenoxy)ethyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
1-[(3-methoxyphenyl)methyl]-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-amine
N-butyl-5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]benzamide
3-[(dimethylamino)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
1-methyl-5-{[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indole
1-{[(3R,4R)-1-(2,5-difluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
1-(2-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,5S,6S)-3-cyclopentyl-N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
1-(1-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
6-methyl-2-{2-[(1-phenoxypropan-2-yl)amino]ethyl}-3,4-dihydropyrimidin-4-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(cyclohexylmethyl)-N-[2-(3-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
2-{1-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
1-(4-phenylazepan-1-yl)-2-(pyrazin-2-yl)ethan-1-one
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-4-(piperidin-3-yl)benzamide
4-(1-{[4-(methoxymethyl)piperidin-1-yl]sulfonyl}piperidin-3-yl)benzoic acid
methyl[(5-methyl-1H-pyrazol-3-yl)methyl]{[2-(trifluoromethyl)phenyl]methyl}amine
2-(1-methylpiperidin-2-yl)-1-(4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-1-yl)ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(dimethyl-1,3-thiazol-5-yl)acetamide
N-cyclobutyl-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1,3-benzothiazole-6-carboxamide
2-[(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]pyrimidine
6-(4-methoxy-3,5-dimethylphenyl)-3,4-dihydroquinazolin-4-one
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-(2-fluorophenyl)ethan-1-one
2-(1-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-amine
4,5-dimethyl 1-[(3S,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
1-(azepan-1-yl)-3-[3-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)acetamide
5-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine