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N-[2-(4-ethylpiperazin-1-yl)-2-methylpropyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
2-(2-butoxy-4-fluorophenyl)-6-(piperidine-1-carbonyl)pyrazine
7-chloro-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
(1S,5R)-3-benzyl-6-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-hydroxy-1-[4-(2-methoxybenzoyl)piperazin-1-yl]-4-(methylsulfanyl)butan-1-one
2-(ethylamino)-4-methyl-N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-1,3-thiazole-5-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-(4-hydroxyphenyl)propanamide
(1S,9R)-11-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)-3-methoxypiperidine
2-{4-chloro-2-[(dimethylamino)methyl]-6-methoxyphenoxy}propanoic acid
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-fluorobenzamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)(pyrazin-2-ylmethyl)amine
N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-(2,6-difluorophenoxymethyl)-N-[2-(methylsulfanyl)ethyl]-1,2-oxazole-3-carboxamide
2-amino-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-6-(1H-indol-3-yl)pyridine-3-carbonitrile
[1-(2H-1,3-benzodioxole-5-carbonyl)-3-(3-phenylpropyl)piperidin-3-yl]methanol
1-ethyl-5-oxo-N-[(1-phenylcyclopentyl)methyl]pyrrolidine-3-carboxamide
3-[1-(4-methoxybenzoyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
8-[(2-butyl-1H-imidazol-4-yl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(prop-2-en-1-ylsulfanyl)propanamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-(1H-pyrazol-1-yl)butanamide
3-[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzonitrile
2-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}propanamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-chloro-5-methylpyridin-2-yl)piperidin-3-ol
N-methyl-N-(1,2-oxazol-3-ylmethyl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(2-hydroxyethyl)-8-(pyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N3-(3-hydroxypropyl)-N1,N1-dimethyl-N3-(pyridin-4-ylmethyl)piperidine-1,3-dicarboxamide
2-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}-2-[4-fluoro-3-(hydroxymethyl)phenyl]acetic acid
1-[(2,6-dimethylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-methyl-N-[2-phenyl-2-(piperidin-1-yl)ethyl]pyridine-3-carboxamide
2-(2,5-dimethoxyphenyl)-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)acetamide
1-cyclobutanecarbonyl-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
5-(2,3-dihydro-1H-inden-1-ylmethyl)-3-propyl-1,2,4-oxadiazole
(3R,4R)-3-methyl-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-4-(oxan-4-yl)piperidin-4-ol
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
(1R,6S)-3-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-9-methyl-3,9-diazabicyclo[4.2.1]nonane
4-{[2-(benzyloxy)phenyl]methyl}-4H-1,2,4-triazole
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[2-(thiophen-3-yl)acetyl]piperidine-4-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
1-{6-[(E)-2-phenylethenyl]pyridin-2-yl}piperazine
4-[4-(adamantan-1-yl)piperazine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetic acid
2-(3-methylbut-2-en-1-yl)-8-(1,3-thiazol-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]acetamide
methyl 2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-6-[(3-methoxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1S,5R)-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
9-(5-methoxyfuran-2-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-({5-[1-(3-methoxypropyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine