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3-[4-(2,7-dimethylquinoline-4-carbonyl)piperazin-1-yl]pyrazine-2-carbonitrile
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
2-(2,3-difluorophenoxymethyl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
(4-{[4-(methylsulfanyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)(pyridin-3-yl)methanol
[(2-ethylpyrimidin-5-yl)methyl][(4-methoxyphenyl)methyl](pyridin-2-ylmethyl)amine
3-(hydroxymethyl)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-ol
8-[2-(4-methylphenoxymethyl)furan-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
3-[2-(methylsulfanyl)benzoyl]-1-(1H-pyrazol-3-ylmethyl)piperidine
2-{5-[(1-methylpyrrolidin-2-yl)methyl]-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-3-yl}acetamide
1-[(2-chloro-6-fluorophenyl)methyl]-4-methyl-1,4-diazepan-5-one
3-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
3-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-5-(phenoxymethyl)-1H-pyrazole
2-(3-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
1-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-4-(hydroxymethyl)piperidin-4-ol
N-cyclopropyl-7-(dimethyl-1,3-thiazole-5-carbonyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-2-(1H-pyrrol-1-yl)propanamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}acetamide
(3S,4R)-3-(dimethylamino)-N-[4-fluoro-3-(trifluoromethyl)phenyl]-4-propylpyrrolidine-1-carboxamide
4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-2-[(3-methoxyphenyl)methyl]morpholine
6-[(3S,4R)-3-acetamido-4-propylpyrrolidin-1-yl]-N-ethyl-N-methylpyridine-3-carboxamide
(4aS,8aS)-2-(2-phenoxyethanesulfonyl)-decahydro-2,7-naphthyridin-4a-ol
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazine
3-(2-ethylbutyl)-8-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-(1-methyl-1H-imidazol-2-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]pyridazin-3-amine
3-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)pyridine
4-{1-[2-(2-methylphenoxy)ethyl]piperidin-4-yl}thiomorpholine
(1R,3s,6r,8S)-4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
2-(2-chloro-4-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)acetamide
(2S,4R)-N-[2-(dimethylamino)ethyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
9-[2-(1H-pyrazol-1-yl)butanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methylphenyl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-3-phenylpropanamide
(3R,4S)-4-cyclopropyl-1-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}pyrrolidin-3-amine
benzyl(cyclobutylmethyl){[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
(3R,4S)-N,N-dimethyl-1-(3-methylpyrazin-2-yl)-4-(propan-2-yl)pyrrolidin-3-amine
9-[(5-propylfuran-2-yl)methyl]-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,5S,6S)-6-[(dimethylamino)methyl]-N-[4-(3-methoxyphenyl)phenyl]-3-azabicyclo[3.1.0]hexane-3-carboxamide
N-{1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]piperidin-4-yl}pyrimidin-2-amine
N-[1-(2-methoxyethyl)-7-(3-phenylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
4-(4-{[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
4-(1H-imidazol-1-ylmethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-ol
N-[(5-{[3-(prop-2-en-1-yloxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
4-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-1-phenylpiperazin-2-one
2-cyclobutyl-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-methyl-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
2-methoxy-1-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepan-1-yl)ethan-1-one
(1S,5R)-6-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(3-methylfuran-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-benzyl-4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1,4-diazepan-6-ol
1-[2-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-2-(thiophen-3-yl)ethan-1-one
8-methoxy-N-[2-(pyrazin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(azepan-1-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}acetamide