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{2-[3-(1-methoxyethyl)phenyl]pyridin-4-yl}methanol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylthiophene-3-carboxamide
4-(hydroxymethyl)-4-(oxan-2-ylmethyl)-N-(2-phenylphenyl)piperidine-1-carboxamide
7-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyrazolo[1,5-a]pyrimidine-6-carboxamide
2-methoxy-N-(2-methoxyethyl)-4-methyl-N-(thiophen-2-ylmethyl)benzamide
5-[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-8-methoxy-2,5-dihydro-1,4-benzoxazepin-3-amine
2-({2-[(cyclobutylformamido)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)benzoic acid
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-{2-[(2R)-2-amino-2-cyclohexylacetamido]-5-methoxyphenyl}-2-methylpropanamide
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-1-benzoxepine-4-carboxamide
3-{3-cyclopentyl-5-[(2-oxo-1,2-dihydropyrimidin-1-yl)methyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
1-cyclopropanecarbonyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidine-4-carboxamide
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
3-[(3S)-3-(dimethylamino)azepane-1-carbonyl]-4-fluorobenzene-1-sulfonamide
ethyl 1-[2-(2-oxopyrrolidin-1-yl)acetyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
3,3,3-trifluoro-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]propanamide
{2-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-1,3-thiazol-4-yl}methanol
N-(1H-imidazol-2-ylmethyl)-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
4-(2-ethoxyphenyl)-3-(4-methyl-1H-imidazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-ethyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}pyrimidine-5-carboxamide
1-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-3-amine
N-{1-[(8-chloro-4-hydroxyquinolin-2-yl)methyl]piperidin-4-yl}methanesulfonamide
N-{4-[(oxolan-2-ylmethyl)carbamoyl]phenyl}-3-(pyridin-3-yl)azetidine-1-carboxamide
1-[(3-fluorophenyl)methyl]-4-{[(3-methyl-1H-indol-2-yl)methyl]amino}pyrrolidin-2-one
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
5-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-(2-phenylethyl)-N-[2-(thiophen-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-(2-ethyl-1H-imidazol-1-yl)propanamide
1-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}piperidin-4-ol
2-amino-2-methyl-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-(cyclopropylmethyl)-9-[(3-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(2-oxo-2-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethyl)imidazolidine-2,4-dione
1-(1-{[(propan-2-yl)carbamoyl]methyl}piperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3,7-dimethyl-11-{5-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-3,7,11-triazaspiro[5.6]dodecane
4-(3-methylpiperidin-1-yl)-3-(4H-1,2,4-triazol-4-yl)benzamide
(benzylsulfamoyl)[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]amine
(4aR,7aS)-1-methyl-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-4-(5-methylfuran-2-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}benzamide
4-({[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]carbamoyl}amino)-N-(2-methoxyethyl)benzamide
1-[2-(2,4-dimethylphenoxy)ethyl]-3-methylimidazolidin-2-one
[(1-benzylpiperidin-4-yl)methyl](methyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
methyl 3-(2,5-difluorobenzoyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2,3-dihydro-1H-inden-2-yl)-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
4-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-1,4-oxazepan-6-ol
N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{4-[(4-ethoxyphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
3-(4-methyl-1H-imidazol-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
3-(difluoromethoxy)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide