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N2-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-N4-methylpyrimidine-2,4-diamine
5-[(4-fluorophenyl)methyl]-5-{1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-3-(2-methoxyethyl)imidazolidine-2,4-dione
1-({5-[(3,4-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]propanamide
2-fluoro-N-{3-oxo-3-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propyl}benzamide
3-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3,4-thiadiazol-2-yl}-1-[1-(pyridin-2-yl)propan-2-yl]urea
N-{1-oxaspiro[4.4]nonan-3-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(4-{4-[(dimethylamino)methyl]phenyl}-3-(hydroxymethyl)phenyl)methanol
1,3-dimethyl-5-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxopyrrolidin-1-yl)acetamide
(1R,6S)-9-methyl-3-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-phenylacetamide
5-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2-methyl-3,4-dihydropyrimidin-4-one
ethyl 1-[1-benzyl-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carbonyl]piperidine-3-carboxylate
5-(2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
8-[(2,6-difluoro-4-methoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
[(6-chloropyridin-3-yl)methyl][(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]methylamine
ethyl 4-oxo-5-phenoxy-1-[2-(1H-1,2,4-triazol-1-yl)propyl]-1,4-dihydropyridine-3-carboxylate
9-[(4-methoxy-3-methylphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
5-({[(2-ethoxyphenyl)methyl](ethyl)amino}methyl)-2-methoxyphenol
N-{[(2S,4S)-4-fluoro-1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]methyl}-2-(3-methoxyphenyl)acetamide
(4aS,8aR)-6-(3-fluoro-4-methoxybenzoyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
2-[1-({1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
8-(5-acetylpyridin-2-yl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(2-chlorophenyl)methyl]-3-[1-(pyridine-2-carbonyl)piperidin-3-yl]propanamide
1-(furan-2-ylmethyl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}piperidine-3-carboxamide
2-[(3S,4R)-3-cyclopropyl-4-(pyridine-2-amido)pyrrolidin-1-yl]acetic acid
2-{[4-(2-methoxyphenyl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-methylbutanamide
3-(3-methoxyphenyl)-1-methyl-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]pyrrolidine-2,5-dione
[(5-chloro-2,3-dimethoxyphenyl)methyl](methyl)[3-(oxolan-2-yl)propyl]amine
2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-6-(piperidine-1-carbonyl)pyrazine
[(3,5-dichloropyridin-4-yl)methyl](1,4-dioxan-2-ylmethyl)methylamine
(4S,6R)-N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-6-methyl-2-sulfanylidene-1,3-diazinane-4-carboxamide
N-(1-benzylpyrrolidin-3-yl)-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
1-(1-methylpiperidin-4-yl)-N-[2-(pyridin-4-yl)ethyl]piperidine-3-carboxamide
N-(2-methylpropyl)-1-[(1s,4s)-4-{[(4-methoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
{1-[(2-aminopyrimidin-5-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
[(2-benzyl-1,3-thiazol-4-yl)methyl](benzylsulfamoyl)amine
N-[4-(4-{[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
1-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-2-(2-hydroxyphenyl)ethan-1-one
1-[(3-hydroxypiperidin-3-yl)methyl]-3-(8-methylquinolin-5-yl)urea
(3S,5S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(2,3,6-trimethylphenoxy)acetamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]isoquinoline-5-carboxamide