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3-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrazine-2-carbonitrile
4-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
N-[(2R)-1-hydroxypropan-2-yl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
(2S,4R)-N-cycloheptyl-1-(3-methylbut-2-en-1-yl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
3-cyclopropyl-5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
4-({1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}amino)-2-methoxypyridine-3-carbonitrile
5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,5R)-3-(3-fluoropyridin-2-yl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(thiophen-2-ylmethyl)propanamide
2-(ethylamino)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrimidine-5-carboxamide
1-(2-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethyl)imidazolidin-2-one
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3-[4-(methylsulfamoyl)phenyl]propanamide
1'-{1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}spiro[indene-1,4'-piperidine]
methyl 6-{[benzyl(methyl)amino]methyl}-3-(5-methylthiophene-2-amido)thieno[2,3-b]pyridine-2-carboxylate
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-1,2-oxazolidine
2-methyl-N-[3-(morpholin-4-yl)propyl]-1-benzofuran-7-carboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-methyl-1-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
1-(1-cyclopentylpiperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-3-yl}propanamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
N-[2-(1-ethylpiperidin-4-yl)ethyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[(3-methylpyridin-4-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
7-(2-hydroxyethyl)-2-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-cyclopentanecarbonyl-N-{[5-(methylcarbamoyl)furan-2-yl]methyl}piperidine-4-carboxamide
(1S,4S)-2-[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-2-azabicyclo[2.2.1]heptane
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-fluorobenzoyl)piperidine
2-{5-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}phenol
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-yl)piperidine
benzyl 4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxylate
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-methyl-N-(quinoxalin-2-ylmethyl)acetamide
1-ethyl-5-{[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
naphthalen-1-yl (7R,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
1-{[4-(butan-2-yloxy)-3-methoxyphenyl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
1-(2-methylphenyl)-4-(6-methylpyridine-2-carbonyl)-1,4-diazepane
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-methyl-1-benzofuran-5-carbonyl)pyrrolidin-3-yl]methanol
(3S,7S,8aS)-3-benzyl-7-({[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(quinolin-2-ylmethyl)benzamide
1-(3-aminoazepan-1-yl)-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
4-(1-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}piperidin-4-yl)thiomorpholine
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-methyl-4-(1-phenyl-1H-pyrazol-5-yl)-1-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-{[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]methyl}-2-methoxyphenol
3-methyl-8-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(1,3-benzothiazol-2-yl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]propanamide
2-[ethyl(pyridin-4-ylmethyl)amino]-2-[4-(propan-2-yloxy)phenyl]acetic acid
[(2S,6S)-4-(pyrazine-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
3-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
6-(3,5-dichloro-2-methoxybenzoyl)-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-{3-tert-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-fluoro-7-methylimidazo[1,2-a]pyridine