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N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
6-methyl-5-[4-(1H-pyrazol-1-yl)phenyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[3-({[1-(1-methyl-1H-pyrazol-5-yl)propyl]carbamoyl}methoxy)phenyl]propanamide
4-[2-(1-ethylpiperidin-4-yl)acetyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
N-(3-fluorophenyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}methanol
5-(2-fluorophenyl)-N-[2-(methylsulfanyl)ethyl]-1,2,4-triazin-3-amine
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-2-(1H-1,2,4-triazol-3-yl)benzamide
2-[cyclopropyl(1H-indol-5-ylmethyl)amino]-N-(1,3-thiazol-2-yl)propanamide
3-(3,4-difluorophenyl)-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]propan-1-one
2-methoxy-6-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)phenol
[1-(2-chlorophenyl)-2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl]dimethylamine
1-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
1-cycloheptyl-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
8-methyl-N-[(5-methylthiophen-2-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-methyl-4-[4-({7-methyl-2,7-diazaspiro[4.4]nonan-2-yl}methyl)phenyl]butan-2-ol
N-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-amine
1-(2-methoxyphenyl)-4-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazin-2-one
3-[(3R)-1-benzylpyrrolidin-3-yl]-1-(3-cyano-4-ethoxyphenyl)-3-methylurea
2-hydroxy-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
2-({4-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
2-(butylsulfanyl)-N4-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}pyrimidine-4,6-diamine
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(hydroxymethyl)piperidin-4-ol
N-benzyl-N-ethyl-3-(3-hydroxy-3-methylbutyl)benzamide
6-chloro-2-(1H-pyrazol-3-yl)quinoline
(1S,9R)-11-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-{2-[3-(1-methylpiperidin-3-yl)propanamido]ethyl}benzoic acid
4-[(2-fluorophenyl)methyl]-1-(2-oxo-2H-chromene-3-carbonyl)-1,4-diazepan-5-one
N-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-phenylpiperidin-4-amine
4-[(2S,4S)-1-(adamantan-2-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]morpholine
N-[2-(methylamino)ethyl]-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(5-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]methanol
(3S,5R)-N3-(4-methylphenyl)-N5-[2-(pyrrolidin-1-yl)ethyl]piperidine-3,5-dicarboxamide
N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(dimethylamino)-8-(4-methanesulfonylphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-cyclobutanecarbonyl-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-4-carboxamide
3-[1-(2-hydroxy-2-phenylethyl)-4-phenyl-1H-imidazol-5-yl]phenol
4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazole
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
methyl (2S)-1-[5-(cyclooctylcarbamoyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carbonyl]pyrrolidine-2-carboxylate
{2-[2-(1H-indol-5-yl)phenoxy]ethyl}dimethylamine
5-{1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}quinoline
2-[(3-{5-[(4-fluoropiperidin-1-yl)methyl]thiophen-2-yl}-1H-pyrazol-1-yl)methyl]-3-methylpyridine
N-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-2,3-dihydro-1H-isoindole-2-carboxamide
N-ethyl-2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyridine-4-carboxamide
3-(5-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}furan-2-yl)-1H-pyrazole
1-(2-aminoethyl)-N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
4-[2-methyl-5-(trifluoromethyl)benzoyl]-1-phenylpiperazin-2-one
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylfuran-2-yl)methyl]acetamide