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3-[(2R,3R,6R)-5-(5-chloropyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
methyl 5-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-5-oxopentanoate
4-[(3-fluoro-4-methylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
2-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)-N-(2,3,4-trifluorophenyl)acetamide
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-[2-(pyridin-3-yl)acetyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5,6-dimethyl-3-[2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-phenylpiperidine-4-carbonitrile
1-{3-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]propyl}pyrrolidin-2-one
N-methyl-2-(4-{pyrazolo[1,5-a]pyridin-7-yl}-1H-pyrazol-1-yl)acetamide
1-(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(4-methoxyphenyl)ethan-1-one
1-(2-fluorobenzoyl)-4-phenoxypiperidine-4-carboxylic acid
(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(4-ethoxy-2-fluorophenyl)urea
3-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]-4-fluorobenzene-1-sulfonamide
3,4,7-trimethyl-2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-1H-indole
(3R,4S)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
(4aS,7aR)-1-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-4-[2-(dimethylamino)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-2-(methylamino)-N-[1-(1,3-thiazol-2-yl)ethyl]pyridine-4-carboxamide
2-(5-{[methyl(thian-4-yl)amino]methyl}furan-2-yl)benzonitrile
4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]-N-(thiophen-3-yl)piperidine-1-carboxamide
2,6,6-trimethyl-3-[2-(4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indol-4-one
2-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)acetamide
2-(ethylamino)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-5-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
2-[(3R,4S)-3-ethanesulfonamido-4-(propan-2-yl)pyrrolidin-1-yl]acetamide
(3S,4S)-1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4-propylpyrrolidine-3-carboxylic acid
2-(3-hydroxypropyl)-8-[(2,3,4-trifluorophenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
7-(cyclobutylmethyl)-2-[(2-phenyl-1,3-oxazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
N-[3-(4-{[2-(3-phenylpyrrolidin-1-yl)ethyl]amino}piperidin-1-yl)phenyl]pyridine-3-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]acetamide
2-(3,4-dichlorophenyl)-4-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]morpholine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-yl)piperidine
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-3-(pyrrolidin-1-yl)piperidine
3-{4-[4-(1-ethoxyethyl)phenyl]-3,5-dimethyl-1H-pyrazol-1-yl}propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-5-methylthiophene-2-carboxamide
1-[(4-fluorophenyl)methyl]-5-(3-methylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(2S,4R)-4-amino-N-ethyl-1-[4-(trifluoromethyl)benzenesulfonyl]pyrrolidine-2-carboxamide
N-(3-hydroxypropyl)-1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
6-{[(dimethylcarbamoyl)methyl]amino}-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
N-{[1-(3-chloro-2-methylbenzenesulfonyl)piperidin-3-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide
5-(dimethylamino)-2-{2-[2-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
(3S,4R)-1-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
(2R,6R)-4-(4-methylpyridine-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
7-(5-methyl-2-phenylfuran-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-(azepan-1-yl)-3-(4-chloro-2-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
2-fluoro-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)benzamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
(3aS,6aR)-5-[(4-hydroxy-3-methylphenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one