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2-[({1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
2-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylformamido}-N,N-dimethyl-2-phenylacetamide
N-(2H-1,3-benzodioxol-5-yl)-1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-3-amine
2-methyl-4-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}quinoline
N-[(2-chlorophenyl)methyl]-5-methyl-N-(propan-2-yl)-1,3,4-oxadiazole-2-carboxamide
8-(2,4-difluorobenzoyl)-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3E)-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]pent-3-en-1-one
4-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-N-ethylmorpholine-2-carboxamide
5-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
8-[(2,6-difluorophenyl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-cyclopropyl-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-6-oxo-1,6-dihydropyridine-3-carboxamide
4-fluoro-3-[3-(pyridin-2-yl)azetidine-1-carbonyl]benzene-1-sulfonamide
N-(1-benzylpiperidin-3-yl)-5-(2-fluorophenyl)-1,2,4-triazin-3-amine
dimethyl({4-methyl-5-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N,N-dimethyl-2-[(1S,5R)-6-[(3-methylquinoxalin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
3-(5-methylfuran-2-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrazole-5-carboxamide
N-{1-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]pyrrolidin-3-yl}-N-methylacetamide
7-(4-fluorophenyl)-2-[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(1S,5R)-3-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1H-indazol-6-yl)-4-[(2R)-oxolane-2-carbonyl]piperazin-2-one
4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-1,3-dimethylpiperazin-2-one
3-methyl-8-[2-(pyridin-3-yl)-1,3-thiazole-4-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methoxy-1-[1'-(3-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-chloro-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)thiophene-2-carboxamide
ethyl 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-({methyl[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-1H-pyrazole-4-carboxylate
3-[(3R,4S)-1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carboxamide
8-(2-methoxyethyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
5-ethyl-2-{4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine
2-chloro-4-{4-[ethyl(methyl)amino]pyrimidin-2-yl}benzamide
8-[(4-fluoro-3-methylphenyl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
4-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperazine-2-carboxylic acid
2-ethyl-4-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-1-methylpiperazine
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2,3-dimethylbenzene-1-sulfonamide
2-(3-chloro-4-fluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(1-methylpiperidin-3-yl)-4-phenylpiperazine
2-{4-[(4-methanesulfonylphenyl)methyl]morpholin-3-yl}acetic acid
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
(1R,2R,6S,7S)-4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[1-(furan-2-carbonyl)piperidin-4-yl]propanamide
(3S,7S,8aS)-3-[(benzyloxy)methyl]-7-{[(2,5-difluorophenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)cyclopropanecarboxamide
(1R,2R,6S,7S)-N-{2-[(dimethylcarbamoyl)methyl]phenyl}-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
1-[2-(furan-2-ylmethoxy)phenyl]-3-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-cyclopropylethan-1-one
(1S,5R)-6-methyl-3-{thieno[3,2-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,5R)-N3-cyclopropyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide