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3-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
3-methyl-N-(1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
N-[(1-methylpiperidin-3-yl)methyl]-2-propylpyridine-4-carboxamide
6-[(3-methoxyphenyl)methoxy]-4-(2-methyl-1,3-thiazole-4-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
2-(2-methoxyphenyl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazine
4-ethyl-6-[3-(2-fluorophenoxy)azetidin-1-yl]-5-methylpyrimidin-2-amine
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-6-(hydroxymethyl)pyridine-2-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)propanamide
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
1-[(2S,4R)-4-[(4-methoxyphenyl)sulfanyl]-1-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
3-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-N,N-dimethylpropanamide
(1S,3R)-3-amino-N-[(5-chloro-2-propoxyphenyl)methyl]cyclopentane-1-carboxamide
(4-{[2-(cyclopentyloxy)phenyl]methyl}morpholin-3-yl)methanol
(3S,9aR)-3-(cyclohexylmethyl)-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4-{[(2S,5R)-5-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)oxolan-2-yl]methyl}phenyl)methanol
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
1-({4-[2-(thiophen-2-yl)azetidine-1-carbonyl]phenyl}methyl)-1H-1,2,3,4-tetrazole
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(2-methylphenyl)-1,4-diazepane-1-carboxamide
2-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)-8-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N,1-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
5-{[(1S)-1-(3-methoxyphenyl)ethyl]carbamoyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrrolidin-3-yl)piperazine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(3-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,4R)-N-ethyl-3-(hydroxymethyl)-N-methyl-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-sulfonamide
2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carboxylic acid
2-{4-[2-(3-methoxyphenyl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
9-(3-fluorobenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(2-methoxyacetamido)-1-methyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
2-benzyl-4-(4-methyl-1,3-oxazole-5-carbonyl)morpholine
(2R,6S)-2,6-dimethyl-4-{1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-yl}morpholine
methyl 2-[({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)(oxolan-2-ylmethyl)sulfamoyl]benzoate
1-[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]piperidin-4-ol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(6-methylpyridine-2-carbonyl)pyrrolidin-3-yl]methanol
7-(1-benzothiophen-3-yl)-4-(pyridazine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(3-cyanophenyl)-3,9-diazaspiro[5.6]dodecane-9-carboxamide
1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
2-(4-{4-[(pyridin-2-ylmethyl)carbamoyl]phenoxy}piperidin-1-yl)acetic acid
N-benzyl-6-(2-phenoxyacetyl)-6-azaspiro[2.5]octane-1-carboxamide
N,5-dimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-[3-(3-methoxyphenoxy)propyl]-4,6-dimethylpyrimidine
5-fluoro-3-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
2-methyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)furan-3-carboxamide
2-phenyl-N-(piperidin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
3-[(methylsulfanyl)methyl]-N-[3-(sulfamoylmethyl)phenyl]piperidine-1-carboxamide
N-cyclopropyl-1-[1-(furan-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide