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methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
N-(4-{[3-methyl-4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)acetamide
4-{2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-benzofuran-5-yl}-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-ol
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(5-methylthiophene-2-carbonyl)pyrrolidin-3-yl]methanol
2-[methyl(pyridin-4-ylmethyl)amino]-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
9-(2-methoxyethyl)-1-methyl-4-(pyridine-2-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(azepan-1-yl)-3-(4-chloro-2-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]{[5-methyl-1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}amine
2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-6-methyl-4H-pyran-4-one
5-(3-methoxy-2,2-dimethylpropanoyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(2S)-2-{[6-(2,5-dimethylfuran-3-yl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
{5-[4-(2,3-dihydro-1H-inden-2-yl)piperazine-1-carbonyl]furan-2-yl}methanol
N-(2,3-dihydro-1H-inden-4-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-(2-methoxyphenoxy)-1-[3-(piperidin-3-yl)benzoyl]piperidine
2,8-dimethyl-4-[3-(2-methylphenyl)piperidine-1-carbonyl]quinoline
4-[1-(1-methylpiperidin-4-yl)-5-(pyridin-2-yl)-1H-1,2,4-triazol-3-yl]benzamide
2-(ethylsulfanyl)-5-({4-[6-(propan-2-yl)pyridin-2-yl]piperazin-1-yl}methyl)pyrimidine
2-(1H-pyrazol-1-yl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]butan-1-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
N-[2-(2-chlorophenyl)ethyl]-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
5-(propan-2-yl)-N-[(1-propyl-1H-imidazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(2-{3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-2-ethyl-1H-imidazole
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(2-fluoro-5-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-{1-[(2,2-difluoro-2H-1,3-benzodioxol-4-yl)methyl]piperidin-4-yl}-2-methyl-3,4-dihydropyrimidin-4-one
1-butyl-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
2-[1-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)azetidin-3-yl]pyridine
N4-[3-(cyclopentyloxy)propyl]-6-methylpyrimidine-2,4-diamine
(1S,9S)-11-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
6-methyl-2-(2-{[1-(2-methylpropyl)piperidin-4-yl]amino}ethyl)-3,4-dihydropyrimidin-4-one
7-(3-chlorophenyl)-4-(3-hydroxypyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
2-methyl-6-(2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)pyrimidin-4-ol
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
8-(5-propyl-1,2,4-oxadiazol-3-yl)-1-oxa-8-azaspiro[4.5]decane
3-amino-1-[(3-ethenylphenyl)methyl]pyrrolidine-3-carboxylic acid
1-(furan-3-carbonyl)-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1,4-diazepane
methyl 5-(2-amino-1,3-benzothiazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
[(5-chlorothiophen-2-yl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
5-(morpholin-4-ylmethyl)-8-[(6-phenylpyridazin-3-yl)oxy]quinoline
3-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
4-(3-methoxyphenyl)-3-[(4-methyl-1,3-thiazol-2-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(2,6-difluorophenoxymethyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-3-carboxamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-4-(1H-pyrazol-3-yl)benzamide
1-methyl-N-[3-(methylsulfanyl)propyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[(4aS,7aR)-4-cyclobutanecarbonyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]pyridine-2-carbonitrile
1-(4-ethylpiperazin-1-yl)-3-[1-(isoquinolin-5-ylmethyl)piperidin-4-yl]propan-1-one
2-[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-1-ium-1-olate
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}(methyl)amino)acetic acid
1-{1-[(4-fluoro-2-methylphenyl)methyl]pyrrolidin-3-yl}piperidine