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N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[(2,3-dimethoxyphenyl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
(4aR,7aS)-1-acetyl-4-[(3-fluorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-ethoxypyridin-3-yl)methyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
2-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
({2-[(2-chlorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)(methyl)(1,3-thiazol-2-ylmethyl)amine
(4aS,7aR)-1-(4-chlorobenzoyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-ethyl-N-(oxolan-2-ylmethyl)acetamide
2-[2-({4-[(dimethylcarbamoyl)methyl]-1,4-diazepan-1-yl}methyl)phenoxy]propanoic acid
N-[2-(1H-imidazol-1-yl)ethyl]-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
(3S,4S)-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinolin-2-yl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
2-[1-(2-methylpropyl)-4-{[4-(trifluoromethoxy)phenyl]methyl}piperazin-2-yl]ethan-1-ol
(3aS,6aS)-1-oxo-2-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4S)-4-amino-1-(2-chloro-5-acetamidobenzoyl)-N,N-diethylpyrrolidine-2-carboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methylpropanamide
2-(3-chloro-4-hydroxyphenyl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
2-amino-1-(2-ethyl-4-{[(1R)-1-phenylethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
N-[(3S,4R)-1-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-4-propylpyrrolidin-3-yl]acetamide
5-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carbonyl}pyridin-2-amine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(1H-pyrazol-1-yl)butanamide
N-(2,3-dihydro-1H-inden-4-yl)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carboxamide
2-ethyl-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1R,3S)-7-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]-7-azaspiro[3.5]nonane-1,3-diol
1-{3-[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]propyl}piperidin-2-one
[1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
(3R,4S)-4-(5-methylfuran-2-yl)-1-phenylmethanesulfonylpyrrolidin-3-amine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(1R,3R)-3-aminocyclopentyl]acetamide
6-[4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carbonyl]-2,3-dimethylquinoxaline
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pyridine-3-carbonyl)pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
3-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
(3aR,7aS)-N-benzyl-N-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-sulfonamide
N-[2-(propylsulfanyl)phenyl]-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
2-({4-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}sulfanyl)ethan-1-ol
1-(butan-2-yl)-N3-cyclohexyl-N3-methyl-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-N-methyl-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[5-({[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]carbamoyl}amino)-2-methylphenyl]propanamide
3-(2-methylpiperidine-1-carbonyl)-N-[2-(pyrazin-2-yl)ethyl]benzene-1-sulfonamide
5-(methoxymethyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1,3,4-oxadiazole-2-carboxamide
N-[3-(carbamoylmethyl)phenyl]-2-[2-(3-hydroxyphenyl)ethyl]piperidine-1-carboxamide
1-[2-(benzenesulfonyl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[4-(2,5-dimethylphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-4-(pyridin-4-yl)-1,4-diazepan-6-ol
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(oxolane-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
1-(3-methoxyphenyl)-3-methyl-4-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]piperazin-2-one
4-{4-[3-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]piperidine-1-carbonyl}benzene-1-sulfonamide
2-(2H-1,3-benzodioxol-5-yloxy)-1-(4-phenyl-1,4-diazepan-1-yl)ethan-1-one
3-{[(1,3-dihydroxypropan-2-yl)amino]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one