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8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-{2-[3-(methanesulfonylmethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(5-ethyl-1,3,4-thiadiazol-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N,N,3,6-tetramethyl-2-[2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-5-yl]quinoline-4-carboxamide
N-[(3R,4S)-1-cycloheptyl-4-cyclopropylpyrrolidin-3-yl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[4-(thian-4-yl)piperazin-1-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
1-[3-(4-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(methylsulfanyl)ethan-1-one
2-{5-[2-(1H-imidazol-2-yl)phenyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl}-6-methylpyridine
(1S,5R)-3-[2-(4-chloro-2-methylphenoxy)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
methyl 3-methyl-4-{[4-(thian-4-yl)piperazine-1-carbonyl]amino}benzoate
5-(2-ethoxyphenyl)pyrimidin-2-amine
N-butyl-2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
2-{1-methyl-5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
4-cyclohexyl-N-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]piperazine-1-carboxamide
(3S,5R)-N3-[(3,4-dimethoxyphenyl)methyl]-N5-(4-fluorophenyl)-1-(pyridin-4-ylmethyl)piperidine-3,5-dicarboxamide
methyl (2S,4S)-4-(2,3-dimethyl-1H-indole-7-amido)-1-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-2-carboxylate
8-cyclobutanecarbonyl-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-(dimethylamino)-2-(4-methylphenyl)-1-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
1-[4-ethoxy-3-(trifluoromethyl)phenyl]-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
(2S)-2-amino-N-(2H-1,3-benzodioxol-5-ylmethyl)-3-methoxy-N-(pentan-3-yl)propanamide
1-[2-(3-methoxyphenyl)azetidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-(2H-1,3-benzodioxol-5-yl)-4-({4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine-1-carboxamide
2-(5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl}-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl)acetic acid
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
N-ethyl-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
2-(2-chlorophenyl)-1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
1-{[1-(2-chlorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}azepan-2-one
N-{[7-(3-chlorothiophene-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}propane-1-sulfonamide
3-(3-acetyl-2-fluorophenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-(1-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
2-{6-hydroxy-4-[2-(methylamino)pyridine-4-carbonyl]-1,4-diazepan-1-yl}acetic acid
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-2-cyclopropyl-1,3-benzoxazole-6-carboxamide
4-{4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazine-1-carbonyl}morpholine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-5-(morpholin-4-ylmethyl)furan-3-carboxamide
ethyl 1-cyclobutyl-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
(cyclohex-3-en-1-ylmethyl)[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]methylamine
3-({1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
(2S,4S)-4-amino-N-ethyl-1-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)sulfonyl]pyrrolidine-2-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[(2-methyl-1H-indol-5-yl)methyl]benzamide
(2S,4R)-N-ethyl-4-(2-hydroxyacetamido)-1-{[2-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carboxamide
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxylic acid
9-(4-fluoro-2-methylbenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
(2E)-N-{[3-methyl-7-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
1-(pyridin-4-yl)-4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperazine